SCHEMBL4787846

SCHEMBL4787846

NC1Cc2c(OCCN3CCCC3)cccc2OC1(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.47
DRD1 P21728 3/20 0.47
DRD4 P21917 3/20 0.47
DRD5 P21918 3/20 0.47
DRD3 P35462 3/20 0.47
DRD2 P14416 2/20 0.46
LTA4H P09960 9/20 0.44
TDP1 Q9NUW8 1/20 0.43
TSHR P16473 1/20 0.42
KDM4E B2RXH2 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750457 0.78 HTR2C (0.41) HRH1KDM4ESMN1; SMN2
SCHEMBL4788942 0.77 GABRA1 (0.34) KDM4E
SCHEMBL4789082 0.73 TDP1 (0.47) HRH1DRD1DRD4DRD5DRD3
Ammonia Solution, Strong SCHEMBL4789081 0.72 TDP1 (0.46) HRH1DRD1DRD4DRD5DRD3
Lithium Ion SCHEMBL4750393 0.67 SIGMAR1 (0.39) DRD2
SCHEMBL4788836 0.66 HRH3 (0.54) DRD3DRD2TDP1TSHRSMN1; SMN2
SCHEMBL7012697 0.65 KDM4E (0.84) HRH1DRD1DRD4DRD5DRD3
SCHEMBL8773745 0.64 HRH1 (1.00) HRH1DRD1DRD4DRD5DRD3
SCHEMBL29573150 0.64 TDP1 (0.66) HRH1DRD1DRD4DRD5DRD3
SCHEMBL30150794 0.64 LTA4H (0.73) HRH1DRD1DRD4DRD5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130319-A2 NOVEL N-TETRAHYDRONAPHTALENE OR N-CHROMANE CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed