SCHEMBL4788693

SCHEMBL4788693

Cc1ccc(C(=O)N2CCc3ccccc3C2)c2c1CC[C@@H](N)C2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.58
ALDH1A1 P00352 2/20 0.58
HTT P42858 2/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
KMT2A Q03164 2/20 0.49
POLB P06746 2/20 0.49
LMNA P02545 1/20 0.49
NOTUM Q6P988 1/20 0.46
BCL2 P10415 2/20 0.45
KDM4E B2RXH2 1/20 0.45
BAD Q92934 1/20 0.45
TSHR P16473 2/20 0.45
HSP90AA1 P07900 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KEAP1 Q14145 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787977 0.83 L3MBTL1 (0.40) HPGDALDH1A1HTTCYP3A4CYP2C9
SCHEMBL4788901 0.77 ALDH1A1 (0.48) HPGDALDH1A1LMNATSHRNPC1
SCHEMBL3456196 0.75 HPGD (1.00) HPGDALDH1A1HTTCYP3A4CYP2C9
SCHEMBL4786769 0.74 KDM4E (0.46) ALDH1A1HTTCYP2C19KMT2APOLB
SCHEMBL14825154 0.72 HPGD (0.79) HPGDALDH1A1HTTCYP3A4CYP2C9
SCHEMBL16588035 0.71 HTT (0.76) HPGDALDH1A1HTTCYP3A4CYP2C9
SCHEMBL7245369 0.68 TSHR (0.37) ALDH1A1HTTKMT2APOLBLMNA
SCHEMBL4212502 0.68 TSHR (0.37) ALDH1A1HTTKMT2APOLBLMNA
SCHEMBL3455489 0.67 HPGD (0.65) HPGDALDH1A1HTTCYP3A4CYP2C9
SCHEMBL11375807 0.67 HPGD (1.00) HPGDALDH1A1HTTCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130319-A2 NOVEL N-TETRAHYDRONAPHTALENE OR N-CHROMANE CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed