SCHEMBL4789169

SCHEMBL4789169

COc1cccc(C2=C(c3ccccc3)C(=O)NC2=O)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.62
PRKCA P17252 4/20 0.62
STK10 O94804 4/20 0.58
SLK Q9H2G2 4/20 0.58
CHEK1 O14757 1/20 0.54
GSK3A P49840 1/20 0.53
NEK2 P51955 1/20 0.53
PTGS2 P35354 2/20 0.53
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3669622 0.85 GSK3B (0.60) GSK3BPRKCASTK10SLKCHEK1
SCHEMBL3822337 0.84 GSK3B (0.69) GSK3BGSK3APTGS2
SCHEMBL5892139 0.81 GAA (0.53) GSK3BPRKCASTK10SLKCHEK1
SCHEMBL114611 0.78 PTGS2 (0.67) GSK3BPTGS2
SCHEMBL18049424 0.77 PTGS2 (0.57) GSK3BPTGS2
SCHEMBL211025 0.77 PDE4B (0.59) GSK3BSTK10SLKPTGS2
SCHEMBL28527835 0.76 MAOA (0.50) GSK3BPRKCASTK10SLKGSK3A
SCHEMBL28080907 0.76 PTGS2 (0.72) GSK3BGSK3APTGS2
SCHEMBL29740761 0.76 CYP1A1 (0.64)
SCHEMBL458391 0.76 CYP1A1 (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO disclosed
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO disclosed