SCHEMBL4789294

SCHEMBL4789294

O=C(O)c1c[nH]c2c(F)cc(Cc3cc(F)cc(C(F)(F)F)c3)cc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
CYP1A2 P05177 2/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.46
ALOX12 P18054 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 1/20 0.45
KDM4E B2RXH2 2/20 0.41
CSNK2A2 P19784 4/20 0.39
CSNK2B P67870 4/20 0.39
CSNK2A1 P68400 4/20 0.39
HSD17B10 Q99714 1/20 0.38
RAB9A P51151 1/20 0.38
TET2 Q6N021 1/20 0.37
TET1 Q8NFU7 1/20 0.37
CMA1 P23946 1/20 0.36
DNA2 P51530 1/20 0.36
CASP6 P55212 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
GPR52 Q9Y2T5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650139 0.90 ALDH1A1 (0.51) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4650802 0.88 ALDH1A1 (0.53) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4650022 0.87 ALDH1A1 (0.50) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4650793 0.83 ALDH1A1 (0.46) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4649289 0.83 ALDH1A1 (0.53) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4650128 0.82 ALDH1A1 (0.52) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4650041 0.81 ALDH1A1 (0.47) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4649447 0.81 RAB9A (0.49) ALDH1A1CYP1A2HPGDLMNAKDM4E
SCHEMBL4649455 0.80 ALDH1A1 (0.50) ALDH1A1CYP1A2HPGDMEN1ALOX12
SCHEMBL4650127 0.79 KDM4A (0.48) ALDH1A1CYP1A2HPGDMEN1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP disclosed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO disclosed