SCHEMBL4790422

SCHEMBL4790422

Oc1ccccc1OC(F)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.43
TP53 P04637 2/20 0.43
TSHR P16473 2/20 0.43
CA1 P00915 1/20 0.43
LMNA P02545 4/20 0.41
MAPT P10636 4/20 0.41
GAA P10253 2/20 0.41
JAK2 O60674 1/20 0.41
AR P10275 1/20 0.36
HSD17B10 Q99714 4/20 0.35
ALOX15 P16050 3/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
KDM4E B2RXH2 2/20 0.35
CYP3A4 P08684 2/20 0.35
NPC1 O15118 1/20 0.35
CA12 O43570 1/20 0.35
GMNN O75496 1/20 0.35
EGFR P00533 1/20 0.35
FYN P06241 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2164883 0.85 ULK1 (0.33) CA2TSHRCA1ALDH1A1CA12
SCHEMBL29118013 0.81 CYP1A2 (0.34) CA2TP53CA1LMNAMAPT
SCHEMBL9095731 0.79 CA1 (0.36) CA2TP53TSHRCA1LMNA
SCHEMBL363528 0.79 CA2 (0.50) CA2TP53TSHRCA1LMNA
SCHEMBL7799614 0.76 ALDH1A1 (0.43) LMNAMAPTGAAALOX15ALDH1A1
SCHEMBL11113864 0.76 ULK1 (0.33)
SCHEMBL8984707 0.76 HTR1A (0.37) CA2TSHRCA1LMNAGAA
SCHEMBL10932877 0.75 CA2 (0.52) CA2TP53TSHRCA1LMNA
SCHEMBL29135349 0.75 CA2 (0.46) CA2TP53TSHRCA1LMNA
SCHEMBL943898 0.74 MEN1 (0.31) MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957495-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-08-20 EP disclosed
WO-2007064045-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-07 WO disclosed
EP-0893444-B1 Process for reparing 2,2,3,3-tetrafluoro-1,4-benzodioxanes, new o-(2-bromo-1,1,2,2,-tetrafluoroethoxy)-phenols and new2-bromo-1,1,2,2-tetrafuoroethoxy-phenylethers LANXESS DEUTSCHLAND GMBH (DE) 2005-11-02 EP disclosed
US-5936102-A CYCLOCONDENSING O-(2-BROMOTETRAFLUOROETHOXY)PHENOL IN THE PRESENCE OF ACID BINDER BAYER AKTIENGESELLSCHAFT (DE) 1999-08-10 US disclosed
EP-0893444-A1 Process for reparing 2,2,3,3-tetrafluoro-1,4-benzodioxanes, new o-(2-bromo-1,1,2,2,-tetrafluoroethoxy)-phenols and new2-bromo-1,1,2,2-tetrafuoroethoxy-phenylethers BAYER AG (DE) 1999-01-27 EP disclosed