SCHEMBL4793607

SCHEMBL4793607

O=S(=O)(c1ccccc1)N1CCN(c2nc(CCCc3ccccc3)cc(-c3ccc(NC4=NCCN4)cc3)n2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.43
CHUK O15111 6/20 0.43
ADRA2A P08913 3/20 0.39
ADRA2B P18089 3/20 0.39
ADRA2C P18825 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HRH1 P35367 1/20 0.36
HRH4 Q9H3N8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4791770 0.92 ADRA2A (0.39) IKBKBCHUKADRA2AADRA2BADRA2C
SCHEMBL4793423 0.86 PIK3CA (0.43) ADRA2AADRA2BADRA2CHTTNPSR1
SCHEMBL4793613 0.82 ITGB3 (0.38) IKBKBCHUKADRA2AADRA2BADRA2C
SCHEMBL4796331 0.76 ADRA2A (0.37) IKBKBCHUKADRA2AADRA2BADRA2C
SCHEMBL4792540 0.76 ADRA2A (0.43) ADRA2AADRA2BADRA2CPTGIRAOC3
SCHEMBL4792493 0.74 PTH1R (0.42) ADRA2AADRA2BADRA2CPTGIRAOC3
SCHEMBL4794483 0.74 PTH1R (0.44) ADRA2AADRA2BADRA2CPTGIRAOC3
SCHEMBL4792633 0.74 PTH1R (0.44) ADRA2AADRA2BADRA2CPTGIRAOC3
SCHEMBL4795789 0.72 ADRA2A (0.39) ADRA2AADRA2BADRA2CPTGIRAOC3
SCHEMBL4906720 0.72 ADRA2A (0.41) ADRA2AADRA2BADRA2CPTGIRAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed