SCHEMBL4796331

SCHEMBL4796331

CN(CCN(C)S(=O)(=O)c1ccccc1)c1nc(CCCc2ccccc2)cc(-c2ccc(NC3=NCCN3)cc2)n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 6/20 0.37
ADRA2B P18089 6/20 0.37
ADRA2C P18825 6/20 0.37
AOC3 Q16853 1/20 0.36
PTGIR P43119 4/20 0.36
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
ITGB3 P05106 2/20 0.35
ITGAV P06756 2/20 0.35
ITGA2B P08514 1/20 0.35
TP53 P04637 1/20 0.35
PTH1R Q03431 2/20 0.34
IKBKB O14920 1/20 0.34
CHUK O15111 1/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4906720 0.86 ADRA2A (0.41) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4795965 0.85 ADRA2A (0.41) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4795892 0.79 ADRA2A (0.41) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4776747 0.79 PKM (0.43) ADORA2AADORA2BADORA1TP53ESR1
SCHEMBL4792540 0.76 ADRA2A (0.43) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4793607 0.76 IKBKB (0.43) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4774170 0.76 PKM (0.41) ADORA2AADORA2BADORA1TP53
SCHEMBL4792493 0.75 PTH1R (0.42) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4791770 0.75 ADRA2A (0.39) ADRA2AADRA2BADRA2CAOC3PTGIR
SCHEMBL4792633 0.74 PTH1R (0.44) ADRA2AADRA2BADRA2CAOC3PTGIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed