SCHEMBL4794075

SCHEMBL4794075

COC(=O)c1cc(Br)n(S(=O)(=O)c2ccccc2)c1.[NaH]

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.55
MEN1 O00255 1/20 0.55
FBP1 P09467 1/20 0.46
KDM4E B2RXH2 3/20 0.44
GAA P10253 3/20 0.44
ALDH1A1 P00352 2/20 0.44
PKM P14618 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 2/20 0.44
PLK1 P53350 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTR6 P50406 1/20 0.42
CTSG P08311 2/20 0.42
CMA1 P23946 2/20 0.42
MAPT P10636 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C1 Q04828 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1156081 0.99 KMT2A (0.56) KMT2AMEN1FBP1KDM4EGAA
SCHEMBL4794078 0.96 KMT2A (0.54) KMT2AMEN1FBP1KDM4EGAA
SCHEMBL1156364 0.86 CYP2C9 (0.46) KMT2AMEN1FBP1KDM4EGAA
SCHEMBL1156214 0.86 ALDH1A1 (0.44) KMT2AMEN1FBP1KDM4EALDH1A1
SCHEMBL1156099 0.85 ALDH1A1 (0.51) FBP1KDM4EGAAALDH1A1TSHR
SCHEMBL1156585 0.85 FBP1 (0.45) KMT2AMEN1FBP1KDM4EALDH1A1
SCHEMBL1156551 0.85 HTR6 (0.43) KMT2AMEN1FBP1KDM4EALDH1A1
SCHEMBL1156490 0.84 ALDH1A1 (0.49) KMT2AMEN1FBP1KDM4EGAA
SCHEMBL5436271 0.79 MEN1 (0.62) KMT2AMEN1FBP1KDM4EGAA
SCHEMBL1156354 0.78 KMT2A (0.49) KMT2AMEN1FBP1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed