SCHEMBL4794147

SCHEMBL4794147

CCOCCOc1nc(CCCc2ccccc2)cc(-c2ccc(NC3=NCCN3)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 8/20 0.40
ADRA2A P08913 11/20 0.39
ADRA2B P18089 10/20 0.39
ADRA2C P18825 10/20 0.39
AOC3 Q16853 1/20 0.37
GPR65 Q8IYL9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4881501 0.91 PTGIR (0.40) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4795011 0.84 PTGIR (0.38) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4793947 0.84 ADRA2A (0.40) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4792540 0.79 ADRA2A (0.43) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4774626 0.79 NOS3 (0.43)
SCHEMBL4795892 0.77 ADRA2A (0.41) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4795965 0.76 ADRA2A (0.41) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4878946 0.76 ADRA2A (0.39) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4792493 0.76 PTH1R (0.42) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL4906720 0.76 ADRA2A (0.41) PTGIRADRA2AADRA2BADRA2CAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed