SCHEMBL4795186

SCHEMBL4795186

COCCN(C(=O)C1CCC(C(F)(F)F)CC1)c1cc(-c2ccc(-c3cc4ncccn4n3)cc2)sc1C(=O)OC

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.35
HTT P42858 1/20 0.35
ATM Q13315 1/20 0.35
PDE4D Q08499 2/20 0.32
SYK P43405 1/20 0.32
NR1H4 Q96RI1 1/20 0.31
RXFP1 Q9HBX9 2/20 0.30
TP53 P04637 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
DGAT1 O75907 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4795177 1.00 ALDH1A1 (0.36) ALDH1A1KDM4EHTTATMPDE4D
SCHEMBL4794178 0.94 ALDH1A1 (0.37) ALDH1A1PDE4DHTR1A
SCHEMBL4794177 0.94 ALDH1A1 (0.37) ALDH1A1PDE4DHTR1A
SCHEMBL4795067 0.92 ALDH1A1 (0.38) ALDH1A1KDM4EHTTATMPDE4D
SCHEMBL4795076 0.92 ALDH1A1 (0.38) ALDH1A1KDM4EHTTATMPDE4D
SCHEMBL4139806 0.86 KDM4E (0.36) KDM4EHTTATMPDE4DSYK
SCHEMBL4139800 0.86 KDM4E (0.36) KDM4EHTTATMPDE4DSYK
SCHEMBL4726527 0.86 ALDH1A1 (0.39) ALDH1A1KDM4ESYKLMNAHPGD
SCHEMBL4726531 0.86 ALDH1A1 (0.39) ALDH1A1KDM4ESYKLMNAHPGD
SCHEMBL4794530 0.85 KDM4E (0.35) ALDH1A1KDM4EHTTATMPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed