SCHEMBL4795240

SCHEMBL4795240

CS(=O)(=O)Nc1cccc(C(=O)c2ncc(Cl)cc2NS(=O)(=O)c2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 5/20 0.48
GPR27 Q9NS67 1/20 0.43
POLB P06746 1/20 0.43
SLC40A1 Q9NP59 2/20 0.43
CCR2 P41597 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CCR4 P51679 1/20 0.41
CCR5 P51681 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PIK3CD O00329 3/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CCR9 P51686 2/20 0.41
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1762607 0.90 CCR9 (0.48) CCR2ALDH1A1KDM4ECCR9
SCHEMBL305792 0.79 CCR9 (0.48) PIK3CGPIK3CDCCR9
SCHEMBL10223070 0.79 CCR9 (0.47) PIK3CDCCR9
SCHEMBL14303638 0.77 CCR9 (0.35) CCR9
SCHEMBL10223574 0.77 HSD17B2 (0.52) CCR2CCR9
SCHEMBL306561 0.76 HSD17B2 (0.51) PIK3CDCCR9
SCHEMBL12594355 0.74 MEN1 (0.47) GPR27CCR2CYP1A2CYP3A4CYP2D6
SCHEMBL4780581 0.74 CCR2 (0.55) GPR27POLBCCR2CYP1A2CYP3A4
SCHEMBL12161743 0.73 LMNA (0.50) GPR27POLBCCR2CYP1A2CYP3A4
SCHEMBL4774906 0.73 KMT2A (0.53) SLC40A1CCR2CYP2C9CCR4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008008431-A2 HETEROARYL SULFONAMIDES AND CCR2/CCR9 CHEMOCENTRYX, INC. (US) 2008-01-17 WO disclosed