SCHEMBL479714

SCHEMBL479714

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(C(=O)O)cc3Cl)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.36
ESRRA P11474 1/20 0.35
FFAR1 O14842 4/20 0.34
TTR P02766 3/20 0.34
MEN1 O00255 1/20 0.34
PPOX P50336 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
CHEK2 O96017 2/20 0.33
PTGER4 P35408 2/20 0.33
PTGER2 P43116 1/20 0.33
HTR2A P28223 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479715 0.93 IGFBP3 (0.35) MRGPRX4FFAR1THRATHRBCHEK2
SCHEMBL480101 0.92 MCL1 (0.35) FFAR1THRATHRBCHEK2PTGER4
SCHEMBL480100 0.88 PTGER4 (0.35) FFAR1PTGER4PTGER2
SCHEMBL479931 0.86 S1PR2 (0.33) TTRMEN1PPOXKMT2ATDP1
SCHEMBL3658320 0.85 AR (0.38) ESRRAFFAR1HTR2ASLC6A4KCNH2
SCHEMBL479983 0.84 KDR (0.36) MEN1KMT2APDK1PDK2PDK3
SCHEMBL733736 0.84 MRGPRX4 (0.35) MRGPRX4ESRRAFFAR1TTRMEN1
SCHEMBL733612 0.84 MRGPRX4 (0.35) MRGPRX4ESRRAFFAR1TTRMEN1
SCHEMBL480761 0.84 MRGPRX4 (0.35) MRGPRX4ESRRAFFAR1TTRMEN1
SCHEMBL480052 0.83 RHEB (0.35) MRGPRX4TTRMEN1PPOXKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed