SCHEMBL479715

SCHEMBL479715

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(C(=O)O)cc3F)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IGFBP3 P17936 2/20 0.35
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
PTGER4 P35408 3/20 0.33
PTGER2 P43116 2/20 0.33
CHEK2 O96017 1/20 0.32
S1PR2 O95136 1/20 0.32
LPAR1 Q92633 1/20 0.32
LPAR5 Q9H1C0 1/20 0.32
FFAR1 O14842 1/20 0.32
HTR2A P28223 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479714 0.93 MRGPRX4 (0.36) PTGER4PTGER2CHEK2FFAR1HTR2A
SCHEMBL480101 0.90 MCL1 (0.35) PTGER4PTGER2CHEK2FFAR1THRA
SCHEMBL480100 0.88 PTGER4 (0.35) PTGER4PTGER2LPAR1LPAR5FFAR1
SCHEMBL479869 0.86 CYP11B1 (0.35) FFAR1HTR2ASLC6A4KCNH2
SCHEMBL480020 0.85 PRKAB2 (0.33) S1PR2
SCHEMBL479931 0.84 S1PR2 (0.33) S1PR2THRATHRB
SCHEMBL480855 0.84 IGFBP3 (0.34) IGFBP3LMNAMAPK1HTTRAB9A
SCHEMBL755674 0.84 IGFBP3 (0.34) IGFBP3LMNAMAPK1HTTRAB9A
SCHEMBL480037 0.83 SCN8A (0.34) FFAR1
SCHEMBL479983 0.83 KDR (0.36) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed