SCHEMBL480100

SCHEMBL480100

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(C(=O)O)cc3)c(Cl)c2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 3/20 0.35
PTGER2 P43116 2/20 0.35
RXRA P19793 1/20 0.34
BRD4 O60885 1/20 0.34
MCL1 Q07820 1/20 0.33
LPAR1 Q92633 5/20 0.33
LPAR5 Q9H1C0 5/20 0.33
FFAR1 O14842 2/20 0.32
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RHEB Q15382 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479998 0.91 ALDH1A1 (0.34) BRD4ALDH1A1
SCHEMBL479197 0.89 SCN8A (0.34) BRD4FFAR1RHEB
SCHEMBL480101 0.88 MCL1 (0.35) PTGER4PTGER2RXRABRD4MCL1
SCHEMBL479715 0.88 IGFBP3 (0.35) PTGER4PTGER2LPAR1LPAR5FFAR1
SCHEMBL479714 0.88 MRGPRX4 (0.36) PTGER4PTGER2FFAR1
SCHEMBL479923 0.84 SCN8A (0.36) FFAR1
SCHEMBL479736 0.83 PTGDR2 (0.35)
SCHEMBL479879 0.82 ACACB (0.32)
SCHEMBL479983 0.80 KDR (0.36) ALDH1A1
SCHEMBL479931 0.80 S1PR2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed