SCHEMBL480084

SCHEMBL480084

Cc1[nH]c(=O)ccc1C(O)(C(C)c1cc(Oc2ccc(C(=O)O)c(Cl)c2)ccc1Cl)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.33
THRA P10827 3/20 0.31
THRB P10828 3/20 0.31
KMO O15229 1/20 0.31
RHEB Q15382 1/20 0.31
FFAR1 O14842 1/20 0.31
EGLN1 Q9GZT9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480149 0.91 KDR (0.32)
SCHEMBL480365 0.86 CYP4F2 (0.37)
SCHEMBL15789678 0.85 MCL1 (0.35) THRATHRBKMORHEBFFAR1
SCHEMBL480092 0.85 PDE2A (0.34)
SCHEMBL480320 0.84 SCN9A (0.34) RHEB
SCHEMBL480107 0.84 KMT2A (0.35)
SCHEMBL480109 0.83 PDK2 (0.36)
SCHEMBL480000 0.80 S1PR2 (0.33) S1PR2THRATHRBKMOFFAR1
SCHEMBL479955 0.78 IGFBP3 (0.35) S1PR2THRATHRBRHEBEGLN1
SCHEMBL480182 0.77 SCN9A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed