SCHEMBL480107

SCHEMBL480107

CCOC(=O)c1cc(Oc2ccc(Cl)c(C(C)C(O)(c3ccc(=O)[nH]c3C)C(F)(F)F)c2)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
MAPT P10636 3/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HTT P42858 1/20 0.31
KDM4E B2RXH2 2/20 0.31
P2RX3 P56373 3/20 0.31
LGALS8 O00214 1/20 0.30
LGALS3 P17931 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480365 0.94 CYP4F2 (0.37) KMT2APDE3BPDE3ACYP1A2CYP4F2
SCHEMBL480149 0.84 KDR (0.32) PDE3BPDE3A
SCHEMBL480084 0.84 S1PR2 (0.33)
SCHEMBL479871 0.82 MRGPRX4 (0.33) KMT2AMEN1HPGDTSHRMAPK1
SCHEMBL754922 0.79 BAZ2B (0.41) CYP1A2MAPTHTTP2RX3CETP
SCHEMBL480108 0.79 BAZ2B (0.41) CYP1A2MAPTHTTP2RX3CETP
SCHEMBL480263 0.79 PPOX (0.33) KMT2AMEN1HPGDNPSR1PDE3B
SCHEMBL480092 0.78 PDE2A (0.34) PDE3BPDE3A
SCHEMBL480172 0.77 NR3C1 (0.34) TSHR
SCHEMBL480155 0.77 SCN8A (0.36) LMNAP2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed