SCHEMBL480263

SCHEMBL480263

CCOC(=O)COc1cc(Oc2ccc(C(C)C(O)(c3ccc(=O)[nH]c3C)C(F)(F)F)c(Cl)c2)ccc1F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPOX P50336 1/20 0.33
DUT P33316 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
ALDH1A1 P00352 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 3/20 0.31
NPSR1 Q6W5P4 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
NTSR1 P30989 1/20 0.31
CYP2C19 P33261 1/20 0.31
P2RX3 P56373 1/20 0.31
PLA2G7 Q13093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480172 0.92 NR3C1 (0.34) TDP1
SCHEMBL754455 0.81 PPOX (0.37) PPOXDUTL3MBTL1GAAPKM
SCHEMBL733146 0.81 PPOX (0.37) PPOXDUTL3MBTL1GAAPKM
SCHEMBL480107 0.79 KMT2A (0.35) L3MBTL1GAAALDH1A1MAPTNPSR1
SCHEMBL480092 0.79 PDE2A (0.34) PDE3BPDE3A
SCHEMBL480171 0.77 CYP11B1 (0.35)
SCHEMBL480365 0.76 CYP4F2 (0.37) L3MBTL1GAAALDH1A1MAPTKMT2A
SCHEMBL479790 0.75 MCL1 (0.36) CYP2C19
SCHEMBL480320 0.74 SCN9A (0.34) PPOXTDP1MEN1KMT2A
SCHEMBL479912 0.73 THRB (0.35) GAAPKMMAPTNPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed