SCHEMBL480139

SCHEMBL480139

COc1ccc(C(C=O)c2ccc(Br)cc2Cl)cn1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
NR3C1 P04150 2/20 0.33
ACLY P53396 1/20 0.33
GPR183 P32249 2/20 0.33
KDM4E B2RXH2 2/20 0.32
PABPC1 P11940 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ERN1 O75460 2/20 0.32
KCNH2 Q12809 1/20 0.32
RECQL P46063 1/20 0.32
NNMT P40261 1/20 0.31
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3630701 0.76 FLT1 (0.35) KMT2ASMN1; SMN2
SCHEMBL480932 0.72 NNMT (0.45) MEN1KMT2ANPC1RAB9AGPR183
SCHEMBL4970732 0.70 MAPT (0.36) MEN1KMT2ARAB9AKDM4EMAOA
SCHEMBL1535156 0.70 NNMT (0.41) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL23539228 0.70 NNMT (0.41) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL31477253 0.68 KMT2A (0.44) MEN1KMT2ANR3C1KDM4EERN1
SCHEMBL5188701 0.67 MAPT (0.44) MEN1KMT2ARAB9AKDM4EKCNH2
SCHEMBL480050 0.67 THRB (0.37) MEN1KMT2ANPC1NR3C1SMN1; SMN2
SCHEMBL34467395 0.66 KMT2A (0.43) MEN1KMT2ANPC1RAB9ANR3C1
SCHEMBL473977 0.66 MAPK1 (0.41) MEN1KMT2AKDM4EERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed