SCHEMBL480183

SCHEMBL480183

COc1cc(-c2ccc(C(C)C(O)(c3c[nH]c(=O)c(C)c3)C(F)(F)F)c(Cl)c2)ccc1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 5/20 0.37
PRKAG1 P54619 5/20 0.37
PRKAA2 P54646 5/20 0.37
PRKAA1 Q13131 5/20 0.37
PRKAG3 Q9UGI9 5/20 0.37
PRKAG2 Q9UGJ0 5/20 0.37
PRKAB1 Q9Y478 5/20 0.37
CHEK1 O14757 1/20 0.36
ESR1 P03372 2/20 0.35
ROCK2 O75116 3/20 0.34
ROCK1 Q13464 3/20 0.34
PIK3CG P48736 1/20 0.34
ADRB3 P13945 3/20 0.33
ADRB1 P08588 2/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RORC P51449 1/20 0.33
MCL1 Q07820 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480057 0.92 CHEK1 (0.37) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479731 0.91 RXRB (0.37) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479963 0.91 PRKAB2 (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480013 0.88 RXRB (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480103 0.88 GRIK1 (0.40) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480079 0.86 PDK2 (0.40) ROCK2ROCK1ALDH1A1
SCHEMBL479948 0.86 ERCC1 (0.36) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479738 0.84 BDKRB1 (0.35)
SCHEMBL479947 0.83 CHEK1 (0.35) CHEK1ROCK2ROCK1
SCHEMBL479931 0.83 S1PR2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed