SCHEMBL4802215

SCHEMBL4802215

CCOc1ccc(N(c2ccc(OCC)cc2)c2nc(N)ncc2F)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.48
SYK P43405 2/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
LMNA P02545 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
TSHR P16473 1/20 0.42
ABCB1 P08183 1/20 0.42
TUBB3 Q13509 1/20 0.42
MAPT P10636 5/20 0.42
NQO1 P15559 1/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 1/20 0.40
GAA P10253 1/20 0.38
MAPK10 P53779 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PKM P14618 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4805497 0.87 KMT2A (0.46) DHFRSYKLMNATSHRABCB1
SCHEMBL27631855 0.87 DHFR (0.40) DHFRSYKSMN1; SMN2LMNAPKM
SCHEMBL27612500 0.84 SYK (0.45) DHFRSYKABCB1TUBB3PKM
SCHEMBL27612476 0.83 SYK (0.43) SYKTDP1MAPTMEN1KMT2A
SCHEMBL27612546 0.82 SYK (0.50) SYKSMN1; SMN2LMNATSHRMAPT
SCHEMBL4802208 0.79 SYK (0.44) DHFRSYKMAPTKDM4EMEN1
SCHEMBL4801168 0.79 SYK (0.54) SYKSMN1; SMN2LMNATDP1TSHR
SCHEMBL27612594 0.78 MAPT (0.49) DHFRSMN1; SMN2LMNATDP1TSHR
SCHEMBL27612831 0.76 RAB9A (0.47) SMN1; SMN2LMNATDP1MAPTHPGD
SCHEMBL4798557 0.75 SYK (0.48) DHFRSYKMAPTKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7329672-B2 2,4-pyrimidinediamine compounds and their uses RIGEL PHARMACEUTICALS, INC. (US) 2008-02-12 US disclosed