SCHEMBL480037

SCHEMBL480037

Cc1cc(C(O)(C(C)c2cc(F)c(Oc3ccc(C(=O)O)c(F)c3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 5/20 0.34
SCN10A Q9Y5Y9 5/20 0.34
SCN9A Q15858 3/20 0.33
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32
MEN1 O00255 1/20 0.32
TTR P02766 1/20 0.32
PPOX P50336 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
FFAR1 O14842 1/20 0.32
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
RHEB Q15382 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479957 0.92 SCN8A (0.36) SCN8ASCN10ASCN9AMET
SCHEMBL480020 0.91 PRKAB2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479915 0.91 PRKAB2 (0.33) SCN9APRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL479197 0.89 SCN8A (0.34) SCN8ASCN10APRKAB2PRKAG1PRKAA2
SCHEMBL479931 0.84 S1PR2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479741 0.84 MET (0.36) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480000 0.84 S1PR2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479715 0.83 IGFBP3 (0.35) FFAR1
SCHEMBL480031 0.83 KMT2A (0.32) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480013 0.83 RXRB (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed