SCHEMBL4810133

SCHEMBL4810133

CC(C)(C)[Si](OCC(=O)Cl)(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 2/20 0.35
CYP3A4 P08684 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PPARA Q07869 2/20 0.34
PPARG P37231 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
HPGD P15428 1/20 0.33
MAPT P10636 2/20 0.33
CYP1A2 P05177 1/20 0.32
ABL1 P00519 1/20 0.32
SLC16A3 O15427 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
CASP3 P42574 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789538 0.86 ALOX15 (0.41) SMYD2CYP3A4HTTSMN1; SMN2CYP2C19
SCHEMBL8354088 0.86 SMYD2 (0.36) SMYD2CYP3A4HTTSMN1; SMN2PPARA
Hydrochloric Acid SCHEMBL29015997 0.86 ALOX15 (0.41) SMYD2CYP3A4HTTSMN1; SMN2CYP2C19
SCHEMBL7336991 0.85 SMYD2 (0.38) SMYD2CYP3A4HTTSMN1; SMN2ALDH1A1
SCHEMBL2030044 0.84 SMYD2 (0.33) SMYD2CYP3A4HTTSMN1; SMN2PPARA
SCHEMBL29102862 0.84 SMYD2 (0.38) SMYD2CYP3A4HTTSMN1; SMN2PPARA
SCHEMBL10828679 0.83 SMYD2 (0.35) SMYD2CYP3A4HTTSMN1; SMN2PPARA
SCHEMBL25712841 0.83 KDM4E (0.39) SMYD2CYP3A4HTTSMN1; SMN2ALDH1A1
SCHEMBL7781357 0.82 POLB (0.39) CYP3A4HTTSMN1; SMN2ALDH1A1HPGD
SCHEMBL26566724 0.82 CYP3A4 (0.37) SMYD2CYP3A4HTTSMN1; SMN2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4694893-A1 NOVEL INHIBITORS OF PIKFYVE AND METHODS USING SAME TME Therapeutics LLC (US) 2026-02-18 EP disclosed
EP-4578860-A1 CYCLOALKYNE DERIVATIVE PeptiDream Inc. (JP) 2025-07-02 EP disclosed
CN-120092006-A Cycloalkyne derivatives 肽梦想株式会社 2025-06-03 CN disclosed
WO-2024216229-A1 NOVEL INHIBITORS OF PIKFYVE AND METHODS USING SAME TME THERAPEUTICS LLC (US) 2024-10-17 WO disclosed
WO-2024043341-A1 CYCLOALKYNE DERIVATIVE ペプチドリーム株式会社 2024-02-29 WO disclosed
CN-110337442-B Novel glucose derivatives as inhibitors of sodium-dependent glucose transporter type 2 东亚ST株式会社 2023-05-12 CN disclosed
US-20170354639-A1 DITERPENOID DERIVATIVES AND METHODS OF USE THEREOF BIOGEN MA INC. 2017-12-14 US disclosed
US-8778974-B2 Trisubstituted 1,2,4 triazoles JANSSEN PHARMACEUTICA NV (BE) 2014-07-15 US disclosed
US-20100324053-A1 TRISUBSTITUTED 1,2,4 TRIAZOLES JANSSEN PHARMACEUTICA NV (BE) 2010-12-23 US disclosed
US-7449468-B2 Thiazole and oxazole derivatives as activators of human peroxisome proliferator activated receptors SMITHKLINE BEECHAM CORPORATION (US) 2008-11-11 US disclosed
US-5300638-A Reacting imine derivative of threonine with an acetyl halide in the presence of a base; preferential BRISTOL-MYERS SQUIBB COMPANY (US) 1994-04-05 US disclosed
EP-0525589-A1 Asymmetric synthesis of taxol side chain Bristol-Myers Squibb Company (US) 1993-02-03 EP disclosed
EP-0154132-B1 6-ALKYLIDENE PENEMS, THEIR PREPARATION AND USE, AND INTERMEDIATES BEECHAM GROUP PLC (GB) 1992-01-08 EP disclosed
EP-0188247-B1 PROCESS FOR PREPARING AZETIDINONE INTERMEDIATES FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-03 EP disclosed
US-4798828-A LACTAMASE INHIBITORS BEECHAM GROUP P.L.C. (GB) 1989-01-17 US disclosed
US-4771134-A Ring-opening process for preparing azetidinone intermediates FARMITALIA CARLO ERBA S.P.A. (IT) 1988-09-13 US disclosed
EP-0232966-A1 Process for the preparation of penem compounds and intermediates for this preparation BEECHAM GROUP PLC (GB) 1987-08-19 EP disclosed
EP-0188247-A1 Process for preparing azetidinone intermediates FARMITALIA CARLO ERBA S.r.l. (IT) 1986-07-23 EP disclosed
EP-0154132-A1 6-Alkylidene penems, their preparation and use, and intermediates BEECHAM GROUP PLC (GB) 1985-09-11 EP disclosed
EP-0120613-A1 Penem derivatives and precursors BEECHAM GROUP PLC (GB) 1984-10-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324053-A1 TRISUBSTITUTED 1,2,4 TRIAZOLES CHRNA1, CHRNA5, CHRNE SMYD2 4308/4885CYP3A4 269/4885HTT 3008/4885
US-20170354639-A1 DITERPENOID DERIVATIVES AND METHODS OF USE THEREOF KEAP1, NFE2L2, HMOX1 SMYD2 4461/4885CYP3A4 1725/4885HTT 61/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.