SCHEMBL4815360

SCHEMBL4815360

CCn1cc(Cc2ccccc2-c2cc(C(=O)NCc3ccccn3)c(OC)cc2C(=O)O)c2ccc(C(=N)NO)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.47
ALDH1A1 P00352 5/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 3/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
HPGD P15428 2/20 0.38
USP2 O75604 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
YWHAG P61981 1/20 0.38
PPARG P37231 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
PIK3CA P42336 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5173183 0.93 PDE10A (0.49) PDE10AALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL4811744 0.85 KMT2A (0.44) PDE10AALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL4811010 0.77 KMT2A (0.44) PDE10AALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL4815144 0.76 PPARG (0.41) PDE10AALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL4812552 0.73 PDE10A (0.42) PDE10AALDH1A1KDM4EKMT2AMEN1
SCHEMBL4805071 0.73 KMT2A (0.44) PDE10AALDH1A1KDM4EKMT2AMEN1
SCHEMBL4809051 0.73 MEN1 (0.44) PDE10AALDH1A1KDM4EKMT2AMEN1
SCHEMBL4811052 0.72 CPT1A (0.39) PPARG
SCHEMBL4809079 0.72 P2RX3 (0.43)
SCHEMBL4808748 0.70 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KDM4EHPGDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7417063-B2 Bicyclic heterocycles useful as serine protease inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-08-26 US claimed