SCHEMBL482340

SCHEMBL482340

Nc1nc2cc(Cl)ccc2s1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.61
IDO1 P14902 1/20 0.61
SMN1; SMN2 Q16637 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
PIK3CD O00329 1/20 0.54
PIK3CA P42336 1/20 0.54
PIK3CB P42338 1/20 0.54
PIK3CG P48736 1/20 0.54
ALDH1A1 P00352 2/20 0.50
TP53 P04637 1/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
EPHX2 P34913 1/20 0.48
HDAC6 Q9UBN7 1/20 0.47
RAB9A P51151 2/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 1/20 0.47
AXL P30530 1/20 0.47
GFER P55789 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29944901 1.00 LOXL2 (0.61) LOXL2IDO1SMN1; SMN2NPSR1PIK3CD
SCHEMBL77839 0.84 RAB9A (0.61) SMN1; SMN2PIK3CDPIK3CAPIK3CBPIK3CG
Hydrochloric Acid SCHEMBL27769376 0.82 RAB9A (0.59) SMN1; SMN2PIK3CDPIK3CAPIK3CBPIK3CG
Hydrochloric Acid SCHEMBL10831817 0.82 RAB9A (0.59) SMN1; SMN2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL780242 0.81 SMN1; SMN2 (0.61) LOXL2IDO1SMN1; SMN2NPSR1ALDH1A1
Nitrogen SCHEMBL29238121 0.81 RAB9A (0.58) SMN1; SMN2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2190447 0.79 ALDH1A1 (0.61) SMN1; SMN2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL7409329 0.78 SMN1; SMN2 (0.58) LOXL2IDO1SMN1; SMN2NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL11236118 0.78 ALDH1A1 (0.59) SMN1; SMN2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL72699 0.76 GAA (0.72) SMN1; SMN2NPSR1PIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398771-A2 HETEROCYCLIC COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2011-12-28 EP claimed
WO-2010096371-A2 HETEROCYCLIC COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-26 WO claimed
EP-1034176-A1 THIOPHENE-SULFONAMIDE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 2000-09-13 EP claimed
WO-1999028316-A1 THIOPHENE-SULFONAMIDE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1999-06-10 WO claimed
JP-7267950-A None JP disclosed
JP-55000344-A None JP disclosed
US-12590071-B2 Hydrazone derivative in which terminal amine group is substituted with aryl group or heteroaryl group, and use thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2026-03-31 US disclosed
US-12545649-B2 WDR5-MYC inhibitors VANDERBILT UNIVERSITY (US) 2026-02-10 US disclosed
CN-120136812-A Compound for targeted degradation of transcription factor KLF5 and application thereof 昆明医科大学 2025-06-13 CN disclosed
WO-2025031129-A1 ARYL UREA DERIVATIVE, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AND USE THEREOF 沈阳药科大学 2025-02-13 WO disclosed
CN-114846013-B Novel aminoaryl derivatives useful as diacylglycerol acyltransferase 2 inhibitors and uses thereof 株式会社LG化学 2024-12-20 CN disclosed
CN-118359602-A Aryl urea derivative and application thereof 沈阳药科大学 2024-07-19 CN disclosed
US-5120872-A Textile dyeing CIBA-GEIGY CORPORATION (US) 1992-06-09 US disclosed
US-4994563-A Dyeing, printing cellulose, silk, wool, synthetic polyamides; colorfastness CIBA-GEIGY CORPORATION (US) 1991-02-19 US disclosed
EP-0349486-A2 Azo dyes, their preparation and their use CIBA-GEIGY AG (CH) 1990-01-03 EP disclosed
US-4236007-A YELLOW SHADES ON POLYESTERS CIBA-GEIGY AKTIENGESELLSCHAFT (CH) 1980-11-25 US disclosed
JP-S55344-A 2-NITROSOIMINOBENZTHIAZOLINE DERIVATIVE IWAKI SEIYAKU KK 1980-01-05 JP disclosed
US-4148805-A POLYESTERS, RED, YELLLOW CIBA-GEIGY AG (CH) 1979-04-10 US disclosed
US-4057638-A Benzothiazole allophanate fungicides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-11-08 US disclosed
US-4041024-A FOR POLYAMIDES AND POLYURETHANES BAYER AKTIENGESELLSCHAFT (DT) 1977-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12545649-B2 WDR5-MYC inhibitors MYC, MYCBP, WDR1 LOXL2 3082/4885IDO1 4396/4885SMN1; SMN2 3142/4885
US-12590071-B2 Hydrazone derivative in which terminal amine group is substituted with aryl group or heteroaryl group, and use thereof ABL1, TH, CYP3A43 LOXL2 1394/4885IDO1 11/4885SMN1; SMN2 4531/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.