SCHEMBL4824911

SCHEMBL4824911

COc1ccc(C(=O)Nc2ccc(S(=O)(=O)NCC(=O)O)cc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.67
LMNA P02545 3/20 0.66
MMP2 P08253 2/20 0.63
MMP9 P14780 1/20 0.63
RAB9A P51151 4/20 0.62
NPC1 O15118 4/20 0.62
TP53 P04637 2/20 0.62
ALOX15 P16050 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
ALDH1A1 P00352 6/20 0.59
MAPT P10636 3/20 0.59
GAA P10253 2/20 0.59
RECQL P46063 1/20 0.59
KMT2A Q03164 4/20 0.58
MEN1 O00255 3/20 0.58
STAT3 P40763 1/20 0.57
MMP3 P08254 1/20 0.57
MMP13 P45452 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
KDM4E B2RXH2 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673498 0.89 LMNA (0.59) HSD17B10LMNARAB9ANPC1SMN1; SMN2
SCHEMBL4173740 0.87 MEP1B (0.67) MMP2MMP9RAB9ANPC1SMN1; SMN2
SCHEMBL7668838 0.86 LMNA (0.68) LMNAMMP2RAB9ANPC1TP53
SCHEMBL5099330 0.86 MEN1 (0.62) HSD17B10LMNAMMP9RAB9ANPC1
SCHEMBL7665894 0.85 LMNA (0.60) LMNAALDH1A1GAAKMT2AMEN1
SCHEMBL7580808 0.85 HSD17B10 (0.61) HSD17B10LMNAMMP2MMP9RAB9A
SCHEMBL7671620 0.84 LMNA (0.59) LMNAALDH1A1GAAKMT2AMEN1
SCHEMBL4834530 0.84 LMNA (0.74) LMNASMN1; SMN2ALDH1A1GAAKMT2A
SCHEMBL7673748 0.84 ALDH1A1 (0.74) LMNASMN1; SMN2ALDH1A1GAAKMT2A
SCHEMBL7663470 0.84 LMNA (0.62) LMNAMMP2SMN1; SMN2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US claimed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP claimed
US-7335686-B2 Method and composition for treating osteoporosis COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-02-26 US disclosed
EP-1678124-A1 NOVEL MOLECULES TO DEVELOP DRUG FOR THE TREATMENT OF OSTEOPOROSIS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-07-12 EP disclosed
WO-2005037774-A1 NOVEL MOLECULES TO DEVELOP DRUG FOR THE TREATMENT OF OSTEOPOROSIS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2005-04-28 WO disclosed
US-20050085537-A1 Method and composition for treating osteoporosis COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-04-21 US disclosed
EP-0757984-B1 Hydroxamic acid derivatives useful for inhibiting gelatinase ONO PHARMACEUTICAL CO (JP) 2002-10-30 EP disclosed
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US disclosed
US-6177466-B1 Sulfonylamino acid derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 2001-01-23 US disclosed
US-6022893-A PREVENTION AND TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION OR EXCESS ACTIVATION OF GELATINASES ONO PHARMACEUTICAL CO., LTD. (JP) 2000-02-08 US disclosed
EP-0757984-A1 Hydroxamic acid derivatives useful for inhibiting gelatinase ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085537-A1 Method and composition for treating osteoporosis SOST, CALCR, MSR1 HSD17B10 2154/4885LMNA 3183/4885MMP2 2736/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.