SCHEMBL4826477

SCHEMBL4826477

O=[N+]([O-])c1cccc(OCC2CC2)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.64
CHRNA4 P43681 2/20 0.64
CHRNB4 P30926 2/20 0.64
CHRNA3 P32297 2/20 0.64
TLR4 O00206 2/20 0.60
TLR2 O60603 2/20 0.60
FAAH O00519 4/20 0.56
SIGMAR1 Q99720 1/20 0.55
SLC6A2 P23975 1/20 0.51
SLC6A4 P31645 1/20 0.51
SLC6A3 Q01959 1/20 0.51
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
CHRNB1 P11230 1/20 0.48
CHRNB3 Q05901 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26378417 0.88 CHRNB4 (0.68) CHRNB2CHRNA4CHRNB4CHRNA3TLR4
SCHEMBL26378416 0.88 CHRNB2 (0.55) CHRNB2CHRNA4CHRNB4CHRNA3TLR4
SCHEMBL15498205 0.87 SLC6A2 (0.58) CHRNB2CHRNA4CHRNB4CHRNA3TLR4
SCHEMBL9239686 0.82 CHRNA3 (0.59) CHRNB2CHRNA4CHRNB4CHRNA3FAAH
SCHEMBL9239680 0.82 CHRNA3 (0.59) CHRNB2CHRNA4CHRNB4CHRNA3FAAH
SCHEMBL4199942 0.82 ALDH1A1 (0.66) CHRNB2CHRNA4CHRNB4CHRNA3FAAH
SCHEMBL4199938 0.82 ALDH1A1 (0.66) CHRNB2CHRNA4CHRNB4CHRNA3FAAH
SCHEMBL4199936 0.82 ALDH1A1 (0.66) CHRNB2CHRNA4CHRNB4CHRNA3FAAH
SCHEMBL3506236 0.81 CHRNB4 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3TLR4
SCHEMBL3506910 0.81 MAPT (0.56) CHRNB2CHRNA4CHRNB4CHRNA3TLR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106946848-A It is used as the derivative of the pyridyl alkyl alcohol of 1 phenyl 2 of phosphodiesterase inhibitors 奇斯药制品公司 2017-07-14 CN disclosed
EP-1948665-A2 THIENOPYRIMIDINONE DERIVATIVES AS MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS Bristol-Myers Squibb Company (US) 2008-07-30 EP disclosed
WO-2007050726-A2 THIENOPYRIMIDINONE DERIVATIVES AS MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-03 WO disclosed