SCHEMBL4826754

SCHEMBL4826754

CNCc1cc(Cl)cc(F)n1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
CD274 Q9NZQ7 1/20 0.34
SLC6A4 P31645 16/20 0.34
HTR2A P28223 13/20 0.34
HTR2C P28335 10/20 0.34
KCNH2 Q12809 6/20 0.33
SLC6A2 P23975 1/20 0.33
TRPV3 Q8NET8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4835449 0.80 KDM4E (0.42) KDM4ETP53CD274SLC6A4HTR2A
SCHEMBL4826581 0.80 NOS3 (0.33) KDM4ETP53SLC6A4HTR2AHTR2C
SCHEMBL26262569 0.77 NOS3 (0.41) KDM4ETP53CD274
SCHEMBL4837374 0.73 KDM4E (0.37) KDM4ETP53SLC6A4HTR2AHTR2C
SCHEMBL24270155 0.72 KDM4E (0.44) KDM4ETP53CD274
SCHEMBL2859978 0.71
SCHEMBL4835923 0.69 KDM4E (0.33) KDM4ETP53SLC6A4HTR2AHTR2C
SCHEMBL12065872 0.69 KDM4E (0.34) KDM4ETP53
SCHEMBL4832258 0.69 KDM4E (0.39) KDM4E
SCHEMBL12536038 0.68 NPSR1 (0.41) KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442692-B2 Indanyl-piperazine compounds LES LABORATOIRES SERVIER (FR) 2008-10-28 US disclosed
WO-2006103342-A9 INDANYL-PIPERAZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2007-10-25 WO disclosed
EP-1707564-B1 Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2007-09-12 EP disclosed
US-20060223830-A1 Indanyl-piperazine compounds LES LABORATOIRES SERVIER (FR) 2006-10-05 US disclosed
EP-1707564-A2 Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2006-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060223830-A1 Indanyl-piperazine compounds HTR4, NR4A1, NR4A3 KDM4E 1559/4885TP53 3984/4885CD274 2158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.