SCHEMBL4828103

SCHEMBL4828103

CN[C@@H]1CCCN(c2cncc(OC)c2)C1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 8/20 0.57
CHRNA4 P43681 8/20 0.57
CHRNB4 P30926 5/20 0.55
CHRNA3 P32297 5/20 0.55
HRH4 Q9H3N8 9/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4827594 1.00 CHRNB2 (0.57) CHRNB2CHRNA4CHRNB4CHRNA3HRH4
SCHEMBL4827593 0.82 CHRNB2 (0.58) CHRNB2CHRNA4CHRNB4CHRNA3HRH4
SCHEMBL4827564 0.82 CHRNB2 (0.58) CHRNB2CHRNA4CHRNB4CHRNA3HRH4
SCHEMBL4819971 0.81 ROCK2 (0.52) HRH4
SCHEMBL4825453 0.81 ROCK2 (0.52) HRH4
SCHEMBL4827811 0.79 ROCK2 (0.56) CHRNB2CHRNA4CHRNB4CHRNA3HRH4
SCHEMBL4821451 0.79 ROCK2 (0.56) CHRNB2CHRNA4CHRNB4CHRNA3HRH4
SCHEMBL30637194 0.78 CHRNB2 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL26106137 0.78 CHRNB2 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL26104729 0.78 CHRNB2 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US claimed
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US disclosed