SCHEMBL4819971

SCHEMBL4819971

CN[C@H]1CCCN(c2cncc(F)c2)C1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.52
ROCK1 Q13464 2/20 0.52
CDC42BPB Q9Y5S2 2/20 0.52
HRH4 Q9H3N8 16/20 0.51
DOT1L Q8TEK3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4825453 1.00 ROCK2 (0.52) ROCK2ROCK1CDC42BPBHRH4DOT1L
SCHEMBL23515071 0.82 KDM4E (0.48)
SCHEMBL4827594 0.81 CHRNB2 (0.57) HRH4
SCHEMBL4828103 0.81 CHRNB2 (0.57) HRH4
SCHEMBL4828087 0.80 HRH4 (0.48) HRH4
SCHEMBL4824732 0.80 CHRNB2 (0.54) ROCK2ROCK1CDC42BPBHRH4
SCHEMBL4830391 0.80 HRH4 (0.48) HRH4
SCHEMBL4823979 0.80 CHRNB2 (0.54) ROCK2ROCK1CDC42BPBHRH4
SCHEMBL4820560 0.79 PIM1 (0.46) HRH4
SCHEMBL4827737 0.79 PIM1 (0.46) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US claimed
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US disclosed