SCHEMBL482849

SCHEMBL482849

CCC([O])N1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HTT P42858 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.33
RECQL P46063 1/20 0.33
USP2 O75604 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
POLB P06746 1/20 0.32
CA12 O43570 1/20 0.32
CA7 P43166 1/20 0.32
CA14 Q9ULX7 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2086387 0.82 TSHR (0.42) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL6539479 0.79 KCNH2 (0.39) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL841129 0.77
SCHEMBL6539704 0.77 KCNH2 (0.39) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL9769982 0.76 ALDH1A1 (0.39) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL3031013 0.76 ALDH1A1 (0.39) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL1994023 0.75 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL1262872 0.75 FDPS (0.36) ALDH1A1MAPTKMT2ANPSR1
SCHEMBL10042012 0.75 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL23108665 0.73 KMT2A (0.42) ALDH1A1LMNAMAPTHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 238 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114555602-B Heterocyclic compounds as STING modulators 百济神州有限公司 2024-02-06 CN claimed
CN-114555602-A Heterocyclic compounds as STING modulators 百济神州有限公司 2022-05-27 CN claimed
WO-2021068866-A1 HETEROCYCLIC COMPOUNDS AS STING MODULATORS BEIGENE, LTD. (KY) 2021-04-15 WO claimed
WO-2007114672-A1 AGENT FOR THE PREVENTION AND TREATMENT OF METABOLIC BONE DISEASE BY ENHANCING OSTEOPROTEGERIN SECRETION OSCOTEC INC. (KR) 2007-10-11 WO claimed
US-6376527-B1 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASES SYNTEX (U.S.A.) LLC 2002-04-23 US claimed
CN-114555602-B Heterocyclic compounds as STING modulators 百济神州有限公司 2024-02-06 CN disclosed
EP-3694856-B1 FUSED TRICYCLIC COMPOUNDS AND USES THEREOF IN MEDICINE SUNSHINE LAKE PHARMA CO LTD (CN) 2023-10-25 EP disclosed
CN-114555602-A Heterocyclic compounds as STING modulators 百济神州有限公司 2022-05-27 CN disclosed
WO-2021068866-A1 HETEROCYCLIC COMPOUNDS AS STING MODULATORS BEIGENE, LTD. (KY) 2021-04-15 WO disclosed
US-10966970-B2 Fused tricyclic compounds and uses thereof in medicine SUNSHINE LAKE PHARMA CO., LTD. (CN) 2021-04-06 US disclosed
EP-3694856-A1 FUSED TRICYCLIC COMPOUNDS AND USES THEREOF IN MEDICINE Sunshine Lake Pharma Co., Ltd. (CN) 2020-08-19 EP disclosed
CN-105732637-B Heteroaromatic compounds and their use in medicine 广东东阳光药业有限公司 2020-04-21 CN disclosed
EP-0724197-A1 Photopolymerizable composition FUJI PHOTO FILM CO., LTD. (JP) 1996-07-31 EP disclosed
EP-0710887-A1 Photopolymerizable composition FUJI PHOTO FILM CO., LTD. (JP) 1996-05-08 EP disclosed
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4138488-A Diphenylmethyl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-06 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10966970-B2 Fused tricyclic compounds and uses thereof in medicine SLC10A1, CYP11B2, CYP11B1 ALDH1A1 1478/4885LMNA 1274/4885MAPT 160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.