Guanine

Guanine

SCHEMBL4830552

Nc1nc2[nH]cnc2c(=O)[nH]1.O=S(=O)(O)O

nearest known ligand 0.53

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Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Guanine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
GLA P06280 1/20 0.53
PMP22 Q01453 1/20 0.53
HSD17B10 Q99714 1/20 0.53
PNP P00491 4/20 0.47
DYRK1A Q13627 1/20 0.42
AKR1B1 P15121 3/20 0.40
MAPT P10636 1/20 0.39
MITF O75030 1/20 0.38
TP53 P04637 1/20 0.38
THRB P10828 1/20 0.38
ALOX15 P16050 1/20 0.38
HBB P68871 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guanine SCHEMBL4658042 0.92 ALDH1A1 (0.61) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL5259 0.92 ALDH1A1 (0.61) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL27542045 0.90 HSD17B10 (0.56) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL9512016 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL21611717 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL865492 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL28373862 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL2895087 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL4063556 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL27400536 0.90 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628558-B1 Process for the synthesis of 9(2-hydroxyethoxy methyl) guanine SOLAR CHEM SA (LU) 1998-04-15 EP claimed
US-5496945-A Process for the synthesis of 9-(2-hydroxyethoxy methyl) guanine SOLAR CHEMICAL S.A. (LU) 1996-03-05 US claimed
EP-0628558-A1 Process for the synthesis of 9(2-hydroxyethoxy methyl) guanine SOLAR CHEMICAL S.A. (LU) 1994-12-14 EP claimed
JP-59027890-A None JP disclosed
CN-112221527-B N, S co-doped porous carbon-coated carbon nanotube bifunctional oxygen electrode catalyst and preparation method thereof 大连理工大学 2021-08-20 CN disclosed
CN-112221527-A N, S co-doped porous carbon-coated carbon nanotube bifunctional oxygen electrode catalyst and preparation method thereof 大连理工大学 2021-01-15 CN disclosed
CN-109502571-A A kind of preparation method of graphene-carbon nano tube composite material 福州大学 2019-03-22 CN disclosed
CN-108864098-A The method that one kind recycling guanine from 2,9- diacetylguanine centrifuge mother liquor 江苏八巨药业有限公司 2018-11-23 CN disclosed
CN-100436590-C Process for producing vitamin B6 DSM IP ASSETS BV (NL) 2008-11-26 CN disclosed
US-20080118926-A1 Method For Detecting Methylation In Genes And Method For Examining Neoplasm Through Detecting Methylation In Genes NATIONAL UNIVERSITY CORPORATION OKAYAMA UNIVERSITY (JP) 2008-05-22 US disclosed
US-7371547-B2 Process for producing vitamin B6 DSM IP ASSETS B.V. (NL) 2008-05-13 US disclosed
EP-1543138-B1 PROCESS FOR PRODUCING VITAMIN B6 DSM IP ASSETS BV (NL) 2006-08-02 EP disclosed
CN-1685052-A Production of vitamin B6Method (2) DSM IP ASSETS BV (NL) 2005-10-19 CN disclosed
EP-1543138-A2 PROCESS FOR PRODUCING VITAMIN B6 DSM IP Assets B.V. (NL) 2005-06-22 EP disclosed
US-20050119411-A1 Polymer composition MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2005-06-02 US disclosed
WO-2004029270-A2 PROCESS FOR PRODUCING VITAMIN B6 DSM IP ASSETS B.V. (NL) 2004-04-08 WO disclosed
EP-0628558-B1 Process for the synthesis of 9(2-hydroxyethoxy methyl) guanine SOLAR CHEM SA (LU) 1998-04-15 EP disclosed
US-5496945-A Process for the synthesis of 9-(2-hydroxyethoxy methyl) guanine SOLAR CHEMICAL S.A. (LU) 1996-03-05 US disclosed
EP-0628558-A1 Process for the synthesis of 9(2-hydroxyethoxy methyl) guanine SOLAR CHEMICAL S.A. (LU) 1994-12-14 EP disclosed
JP-S5927890-A PURIFICATION OF GUANINE KOHJIN CO LTD 1984-02-14 JP disclosed