SCHEMBL483647

SCHEMBL483647

c1ccc(-c2cccc3c2Cc2ccccc2-3)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.46
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
KDM4E B2RXH2 5/20 0.45
LMNA P02545 3/20 0.45
CCR1 P32246 2/20 0.45
CCR5 P51681 2/20 0.45
CCR8 P51685 2/20 0.45
CYP1A2 P05177 2/20 0.45
POLB P06746 1/20 0.45
METAP1 P53582 1/20 0.45
BLM P54132 1/20 0.45
HIF1A Q16665 1/20 0.45
DOHH Q9BU89 1/20 0.45
P4HTM Q9NXG6 1/20 0.45
TP53 P04637 3/20 0.44
ALOX15 P16050 2/20 0.44
HTT P42858 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5934925 0.95 PNMT (0.45) PNMTDRD2DRD4DRD3KDM4E
SCHEMBL28843845 0.87 DRD2 (0.42) PNMTDRD2DRD4DRD3KDM4E
Fluorene SCHEMBL27530322 0.85 KDM4E (0.52) KDM4ELMNACCR1CCR5CCR8
Fluorene SCHEMBL27950409 0.83 KDM4E (0.61) KDM4ELMNACCR1CCR5CCR8
SCHEMBL31443024 0.81 PNMT (0.49) PNMTDRD2DRD4DRD3KDM4E
SCHEMBL30103334 0.80 PNMT (0.63) PNMTDRD2DRD4DRD3KDM4E
SCHEMBL524602 0.80 PNMT (0.63) PNMTDRD2DRD4DRD3KDM4E
SCHEMBL26402107 0.79 UCHL1 (0.43) DRD2KDM4ELMNACCR1CCR5
SCHEMBL9988299 0.78 PNMT (0.42) PNMTDRD2DRD4DRD3NPC1
SCHEMBL2877998 0.78 PNMT (0.61) PNMTDRD2DRD4DRD3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 174 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499181-B1 POLYMER FOR OPTOELECTRONIC DEVICE BOE TECHNOLOGY GROUP CO LTD (CN) 2020-05-13 EP claimed
EP-2139929-B1 POLYCARBAZOLYL(METH)ACRYLATE LIGHT EMISSIVE COMPOSITIONS GEN ELECTRIC (US) 2014-10-08 EP claimed
US-8512879-B2 Polymer for optoelectronic device GENERAL ELECTRIC COMPANY (US) 2013-08-20 US claimed
EP-2499181-A1 POLYMER FOR OPTOELECTRONIC DEVICE General Electric Company (US) 2012-09-19 EP claimed
US-7973126-B2 Emissive polymeric materials for optoelectronic devices GENERAL ELECTRIC COMPANY (US) 2011-07-05 US claimed
WO-2011059553-A1 POLYMER FOR OPTOELECTRONIC DEVICE GENERAL ELECTRIC COMPANY (US) 2011-05-19 WO claimed
US-20110108807-A1 POLYMER FOR OPTOELECTRONIC DEVICE GENERAL ELECTRIC COMPANY (US) 2011-05-12 US claimed
US-7830081-B2 Optoelectronic devices with multilayered structures GENERAL ELECTRIC COMPANY (US) 2010-11-09 US claimed
EP-2225346-A1 EMISSIVE POLYMERIC MATERIALS FOR OPTOELECTRONIC DEVICES General Electric Company (US) 2010-09-08 EP claimed
EP-2162457-A2 CARBAZOLYL POLYMERS FOR ORGANIC ELECTRONIC DEVICES General Electric Company (US) 2010-03-17 EP claimed
WO-2008130806-A1 POLYCARBAZOLYL(METH)ACRYLATE LIGHT EMISSIVE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2008-10-30 WO claimed
US-20080258111-A1 POLYCARBAZOLYL(METH)ACRYLATE LIGHT EMISSIVE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2008-10-23 US claimed
US-20080262184-A1 POLYCARBAZOLYL(METH)ACRYLATE LIGHT EMISSIVE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2008-10-23 US claimed
EP-1963925-A2 LONG LIFE PHOTOCONDUCTORS Lexmark International, Inc. (US) 2008-09-03 EP claimed
US-20080135806-A1 CARBAZOLYL POLYMERS FOR ORGANIC ELECTRONIC DEVICES GENERAL ELECTRIC COMPANY (US) 2008-06-12 US claimed
US-20070225464-A1 OPTOELECTRONIC DEVICES WITH MULTILAYERED STRUCTURES GENERAL ELECTRIC COMPANY (US) 2007-09-27 US claimed
WO-2007070493-A2 LONG LIFE PHOTOCONDUCTORS LEXMARK INTERNATIONAL, INC. (US) 2007-06-21 WO claimed
US-20070134570-A1 Long life photoconductors LEXMARK INTERNATIONAL, INC. 2007-06-14 US claimed
US-6432597-B1 CHARGE GENERATING COMPOUND, CHARGE TRANSFER COMPOUND LEXMARK INTERNATIONAL, INC. 2002-08-13 US claimed
US-6004708-A PHOTOCONDUCTOR USED IN ELECTROPHOTOGRAPHIC REPRODUCTION DEVICES HAVING CHARGE GENERATING LAYER AND CHARGE TRANSPORT LAYER WHICH EXHIBITS REDUCED ROOM LIGHT AND CYCLING FATIGUE WITHOUT NEGATIVELY IMPACTING ON SENSITIVITY LEXMARK INTERNATIONAL, INC. (US) 1999-12-21 US claimed