SCHEMBL4841759

SCHEMBL4841759

CC(N)(Nc1nc(Oc2ccc(F)cc2)nc2[nH]nc(-c3ccccc3Cl)c12)S(N)(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.34
PTGS1 P23219 1/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
DGAT2 Q96PD7 3/20 0.31
PDE2A O00408 1/20 0.31
PDE10A Q9Y233 1/20 0.31
MAPT P10636 1/20 0.31
SCN9A Q15858 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30
CCR4 P51679 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4842636 0.82 DGAT2 (0.33) PTGS2PTGS1L3MBTL1DGAT2PDE2A
SCHEMBL4841715 0.80 DGAT2 (0.32) PTGS2PTGS1L3MBTL1DGAT2PDE2A
SCHEMBL4841726 0.80 DGAT2 (0.36) PTGS2PTGS1L3MBTL1DGAT2
SCHEMBL4842631 0.80 L3MBTL1 (0.34) PTGS2L3MBTL1DGAT2PDE2APDE10A
SCHEMBL4837740 0.80 SCN9A (0.36) CNR1CNR2DGAT2PDE2APDE10A
SCHEMBL14018946 0.76 SCN9A (0.34) DGAT2PDE2APDE10ASCN9A
SCHEMBL4833086 0.76 SCN9A (0.34) DGAT2PDE2APDE10ASCN9A
SCHEMBL4845291 0.72 MAPK14 (0.39) CNR1CNR2DGAT2
SCHEMBL4841381 0.72 MAPK14 (0.40) CNR1CNR2DGAT2
SCHEMBL14018955 0.72 MAPK14 (0.44) PTGS2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435731-B2 Substituted pyrazolo[3,4-d]pyrimadines and methods of using the same ROCHE PALO ALTO LLC (US) 2008-10-14 US disclosed