SCHEMBL4846119

SCHEMBL4846119

CN(C)CCOc1ccc(-c2c(F)cccc2F)cc1C=CC(=O)c1ccccc1CN(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
HRH1 P35367 1/20 0.39
SLC6A9 P48067 1/20 0.38
PADI4 Q9UM07 1/20 0.38
BCHE P06276 2/20 0.37
ACHE P22303 2/20 0.37
PTPN1 P18031 1/20 0.37
KDR P35968 2/20 0.37
RXFP1 Q9HBX9 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAOB P27338 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAOA P21397 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
MCHR1 Q99705 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847346 0.90 KDM4E (0.39) KDM4EHRH1SLC6A9PADI4BCHE
SCHEMBL4846112 0.90 KDM4E (0.39) KDM4EHRH1SLC6A9PADI4BCHE
SCHEMBL4846157 0.89 BCHE (0.42) KDM4EHRH1BCHEACHEPTPN1
SCHEMBL4853004 0.89 HRH3 (0.40) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4847882 0.87 HRH1 (0.39) KDM4EHRH1BCHEACHEPTPN1
SCHEMBL4850158 0.86 SLC6A9 (0.41) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4854570 0.86 HRH1 (0.41) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4851092 0.85 ALDH1A1 (0.42) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4852988 0.85 HRH1 (0.41) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4848073 0.84 HTR7 (0.41) KDM4EHRH1SLC6A9BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed