SCHEMBL4846982

SCHEMBL4846982

NC(=O)c1ccc2c(c1)N=Cc1c(cccc1-c1ccc(F)cc1)N2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.45
CHEK2 O96017 3/20 0.40
FYN P06241 1/20 0.39
CCNE2 O96020 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
MKNK2 Q9HBH9 2/20 0.38
KIT P10721 2/20 0.38
GAK O14976 1/20 0.38
PDGFRB P09619 1/20 0.38
FLT3 P36888 1/20 0.38
MARK1 Q9P0L2 1/20 0.38
STK17A Q9UEE5 1/20 0.38
PTGS1 P23219 1/20 0.38
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
PARP1 P09874 1/20 0.38
GRM2 Q14416 2/20 0.37
MKNK1 Q9BUB5 1/20 0.37
ABL1 P00519 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554153 0.69 HPGDS (0.44) CNR1CHEK2FYNCDK2PARP1
SCHEMBL30131529 0.66 PTGS1 (0.54) CHEK2MKNK2KITGAKPDGFRB
SCHEMBL28203139 0.64 PTGS1 (0.53) CHEK2MKNK2KITGAKPDGFRB
SCHEMBL1290758 0.64 SIRT2 (0.36) CHEK2CCNE2CCNE1CDK2MKNK2
SCHEMBL1926791 0.64 PARP1 (0.63) CHEK2FLT3PARP1
SCHEMBL18165201 0.63 MAPK14 (0.52) CHEK2MKNK2PTGS1PARP1GRM2
Hydrochloric Acid SCHEMBL18152459 0.63 PTGS1 (0.48) CHEK2MKNK2KITGAKPDGFRB
SCHEMBL1132587 0.63 TRPA1 (0.40)
SCHEMBL12056910 0.62 SIRT2 (0.50) PARP1ABL1
SCHEMBL1927476 0.62 BCL2L1 (0.64) CHEK2MKNK2KITGAKPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937677-A1 CB-1 MODULATING COMPOUNDS AND THEIR USE Arcadia Pharmaceuticals Inc. (US) 2008-07-02 EP disclosed
WO-2007047737-A1 CB-1 MODULATING COMPOUNDS AND THEIR USE ACADIA PHARMACEUTICALS INC. (US) 2007-04-26 WO disclosed