SCHEMBL4847640

SCHEMBL4847640

Nc1ccc(OC(F)(F)F)cc1C(=O)NCC(=O)N[C@@H]1CCNC1

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 18/20 0.61
CCR3 P51677 1/20 0.50
HTR2C P28335 1/20 0.46
EPHX1 P07099 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4849796 1.00 CCR2 (0.61) CCR2CCR3HTR2CEPHX1
Acetic Acid SCHEMBL5702355 0.96 CCR2 (0.57) CCR2CCR3HTR2CEPHX1
Acetic Acid SCHEMBL5702362 0.96 CCR2 (0.57) CCR2CCR3HTR2CEPHX1
Nitric Acid SCHEMBL5268270 0.95 CCR2 (0.57) CCR2CCR3HTR2CEPHX1
Nitric Acid SCHEMBL5268257 0.95 CCR2 (0.57) CCR2CCR3HTR2CEPHX1
SCHEMBL4846680 0.85 CCR2 (0.66) CCR2CCR3
SCHEMBL4846664 0.85 CCR2 (0.66) CCR2CCR3
SCHEMBL4839283 0.82 CCR2 (0.49) CCR2CCR3HTR2CEPHX1
SCHEMBL5449234 0.82 CCR2 (0.49) CCR2CCR3HTR2CEPHX1
SCHEMBL27542093 0.78 CCR2 (0.57) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100418951-C Cycloamine derivative and its use as medicine TEIJIN KASEI LTD (JP) 2008-09-17 CN disclosed
US-7390830-B1 Remedies or prophylactics for diseases in association with chemokines TEIJIN LIMITED (JP) 2008-06-24 US disclosed
US-20070249847-A1 Method for Producing Acetamidopyrrolidine Derivatives and Intermediate Compounds Thereof TEIJIN PHARMA LIMITED (JP) 2007-10-25 US disclosed
US-20070249847-A1 Method for Producing Acetamidopyrrolidine Derivatives and Intermediate Compounds Thereof TEIJIN PHARMA LIMITED (JP) 2007-10-25 US disclosed
US-20070249847-A1 Method for Producing Acetamidopyrrolidine Derivatives and Intermediate Compounds Thereof TEIJIN PHARMA LIMITED (JP) 2007-10-25 US disclosed
EP-1760075-A1 METHOD FOR PRODUCING ACETAMIDOPYRROLIDINE DERIVATIVE AND INTERMEDIATE COMPOUND THEREOF Teijin Pharma Limited (JP) 2007-03-07 EP disclosed
EP-1760075-A1 METHOD FOR PRODUCING ACETAMIDOPYRROLIDINE DERIVATIVE AND INTERMEDIATE COMPOUND THEREOF Teijin Pharma Limited (JP) 2007-03-07 EP disclosed
CN-1240699-C Therapeutic or prophylactic agent for chemokine-associated diseases TEIJIN LTD (JP) 2006-02-08 CN disclosed
EP-1179341-B1 REMEDIES OR PREVENTIVES FOR DISEASES IN ASSOCIATION WITH CHEMOKINES TEIJIN LTD (JP) 2005-11-09 EP disclosed
CN-1660815-A Cyclic amine derivatives and their use as drugs TEIJIN LTD (JP) 2005-08-31 CN disclosed
EP-1553085-A1 Cyclic amine derivatives and their use as drugs TEIJIN LIMITED (JP) 2005-07-13 EP disclosed
EP-1535909-A2 Cyclic amine derivatives and their use as drugs TEIJIN LIMITED (JP) 2005-06-01 EP disclosed
CN-1496981-A Cyclic amine derivatives and their use as pharmaceuticals ������������ʽ���� 2004-05-19 CN disclosed
CN-1384743-A Remedies or preventives for diseases in association with chemokines TEIJIN LTD (JP) 2002-12-11 CN disclosed
US-6451842-B1 Cyclic amine derivatives and their use as drugs DUPONT PHARMACEUTICALS COMPANY 2002-09-17 US disclosed
US-6410566-B1 ATHEROSCLEROSIS; ANTIARTHRITIC AGENTS TEIJIN LIMITED (JP) 2002-06-25 US disclosed
US-6362177-B1 INHIBITION OF CHEMOKINE BINDING TEIJIN LIMITED (JP) 2002-03-26 US disclosed
EP-1179341-A1 REMEDIES OR PREVENTIVES FOR DISEASES IN ASSOCIATION WITH CHEMOKINES TEIJIN LIMITED (JP) 2002-02-13 EP disclosed
CN-1279668-A Cyclic amine derivatives and their use as pharmaceuticals TEIJIN LTD (JP) 2001-01-10 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249847-A1 Method for Producing Acetamidopyrrolidine Derivatives and Intermediate Compounds Thereof HDHD5, CBR3, ADH5 CCR2 1243/4885CCR3 1225/4885HTR2C 2802/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.