SCHEMBL4847755

SCHEMBL4847755

COc1ccc(C(=O)C=Cc2cc(-c3cc(C)cc(C)c3)ccc2OCCN(C)C)cc1F

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 9/20 0.46
RELA Q04206 2/20 0.42
ABCG2 Q9UNQ0 2/20 0.42
MCHR1 Q99705 1/20 0.41
CAPN1 P07384 1/20 0.41
SNCA P37840 1/20 0.41
TUBB1 Q9H4B7 1/20 0.41
PTPN1 P18031 1/20 0.41
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847320 0.91 SNCA (0.44) TNFRSF1ASNCAPTPN1THRATHRB
SCHEMBL4847832 0.89 ABCG2 (0.46) TNFRSF1AABCG2CAPN1SNCATUBB1
SCHEMBL4847433 0.89 TNFRSF1A (0.46) TNFRSF1AABCG2MCHR1CAPN1SNCA
SCHEMBL4856242 0.88 BCHE (0.45) TNFRSF1ARELAABCG2
SCHEMBL6386830 0.87 ABCG2 (0.52) TNFRSF1AABCG2PTPN1
SCHEMBL4853345 0.86 RELA (0.48) TNFRSF1ARELAPTPN1
SCHEMBL4852218 0.85 CAPN1 (0.50) TNFRSF1ACAPN1PTPN1
SCHEMBL4849986 0.85 BCHE (0.46) TNFRSF1AABCG2CAPN1PTPN1
SCHEMBL14280884 0.85 BCHE (0.46) TNFRSF1AABCG2CAPN1PTPN1
SCHEMBL4849921 0.84 BCHE (0.45) TNFRSF1APTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed