SCHEMBL4849762

SCHEMBL4849762

CN(C)CCOc1ccc(C(C)(C)C)cc1C=CC(=O)c1ccc(O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
CAPN1 P07384 1/20 0.52
BCHE P06276 1/20 0.47
ACHE P22303 1/20 0.47
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PTPN1 P18031 6/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1B1 Q16678 1/20 0.46
DPP4 P27487 4/20 0.46
IDH1 O75874 1/20 0.45
ABCB1 P08183 1/20 0.45
UGT1A1 P22309 1/20 0.45
ABCC1 P33527 1/20 0.45
PRMT6 Q96LA8 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854287 0.90 PTPN1 (0.55) CAPN1BCHEACHECTSLCTSB
SCHEMBL4854982 0.87 KDM4E (0.47) KDM4EBCHEACHEPTPN1CYP1A1
SCHEMBL4852544 0.85 KDM4E (0.47) KDM4ECAPN1PTPN1CYP1A1CYP1B1
SCHEMBL4849818 0.82 KDM4E (0.51) KDM4ECAPN1BCHEACHELMNA
SCHEMBL4848121 0.82 BCHE (0.55) KDM4ECAPN1BCHEACHECTSL
SCHEMBL4849756 0.82 KDM4E (0.51) KDM4ECAPN1BCHEACHELMNA
SCHEMBL4852218 0.81 CAPN1 (0.50) CAPN1BCHEACHECTSLCTSB
SCHEMBL7186672 0.80 CYP1A1 (0.50) CAPN1PTPN1CYP1A1CYP1B1DPP4
SCHEMBL4855894 0.79 KDM4E (0.48) KDM4EBCHEACHECYP1A1CYP1B1
SCHEMBL7179055 0.79 LMNA (0.49) KDM4ECAPN1PTPN1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed