SCHEMBL4848635

SCHEMBL4848635

CC1CN(c2ncc(CO)cc2Cl)CCN1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.43
BCL2A1 Q16548 2/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
KIT P10721 1/20 0.38
CXCR3 P49682 1/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
XIAP P98170 1/20 0.36
BIRC2 Q13490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2418856 1.00 HRH4 (0.43) HRH4BCL2A1ALDH1A1LMNAADRA2A
SCHEMBL18901972 0.90 HRH4 (0.41) HRH4BCL2A1ALDH1A1LMNAADRA2A
SCHEMBL2417605 0.85 HRH4 (0.41) HRH4BCL2A1ALDH1A1LMNAKIT
SCHEMBL2421495 0.83 CXCR3 (0.41) HRH4BCL2A1CXCR3
SCHEMBL2422155 0.82 HRH4 (0.55) HRH4BCL2A1ALDH1A1LMNAKIT
SCHEMBL2417945 0.82 CXCR3 (0.41) CXCR3
SCHEMBL2420637 0.82 CXCR3 (0.40) HRH4BCL2A1ALDH1A1LMNACXCR3
SCHEMBL899509 0.81 USP28 (0.43)
SCHEMBL907759 0.80 HRH4 (0.45) HRH4BCL2A1ALDH1A1LMNAKIT
SCHEMBL907761 0.80 HRH4 (0.45) HRH4BCL2A1ALDH1A1LMNAKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439360-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2008-10-21 US disclosed
US-20060084640-A1 Vanilloid receptor ligands and their use in treatments AMGEN INC. 2006-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084640-A1 Vanilloid receptor ligands and their use in treatments TRPV1, TRPV3, TRPV2 HRH4 13/4885BCL2A1 2099/4885ALDH1A1 2416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.