SCHEMBL484938

SCHEMBL484938

CC(C)(C)OC(=O)N1CCCC2(CCCNC2)C1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
HSD17B10 Q99714 1/20 0.43
NAMPT P43490 5/20 0.41
HPGD P15428 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP3A4 P08684 3/20 0.39
USP2 O75604 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP11B2 P19099 1/20 0.38
ACACB O00763 2/20 0.38
SCD5 Q86SK9 1/20 0.37
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL484745 0.94 ALDH1A1 (0.50) ALDH1A1HSD17B10NAMPTCYP1A2CYP2C9
SCHEMBL30248648 0.94 CYP3A4 (0.41) ALDH1A1HSD17B10NAMPTHPGDCYP1A2
SCHEMBL484405 0.94 CYP3A4 (0.41) ALDH1A1HSD17B10NAMPTHPGDCYP1A2
SCHEMBL18686085 0.94 CYP3A4 (0.41) ALDH1A1HSD17B10NAMPTHPGDCYP1A2
Hydrochloric Acid SCHEMBL5322449 0.93 ALDH1A1 (0.49) ALDH1A1HSD17B10NAMPTCYP1A2CYP2C9
Oxalic Acid SCHEMBL29782913 0.91 HSD17B10 (0.49) ALDH1A1HSD17B10NAMPTCYP1A2CYP2C9
SCHEMBL2177880 0.90 HPGD (0.42) ALDH1A1HSD17B10HPGDCYP1A2CYP2C9
SCHEMBL14801521 0.90 ALDH1A1 (0.42) ALDH1A1HSD17B10NAMPTHPGDCYP3A4
Hydrochloric Acid SCHEMBL20512854 0.89 HPGD (0.41) ALDH1A1HPGDCYP1A2CYP2C9CYP2D6
SCHEMBL18047957 0.87 USP2 (0.41) ALDH1A1HPGDUSP2SMN1; SMN2CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250276981-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. 2025-09-04 US disclosed
EP-4536650-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. (US) 2025-04-16 EP disclosed
WO-2025039676-A1 PAN-KRAS PROTEIN TARGETED DEGRADER COMPOUND AND USE THEREOF 贝达药业股份有限公司 2025-02-27 WO disclosed
CN-119317623-A Tricyclic quinolone BCL6 bifunctional degradation agents 树线生物科学公司 2025-01-14 CN disclosed
EP-3743425-B1 2,8-DIACYL-2,8-DIAZASPIRO[5.5]UNDECANE COMPOUNDS USEFUL AS IMMUNOMODULATORS BRISTOL MYERS SQUIBB CO (US) 2024-11-27 EP disclosed
US-20240287091-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. 2024-08-29 US disclosed
WO-2023240038-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. (US) 2023-12-14 WO disclosed
CN-111793077-B PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 东莞市东阳光新药研发有限公司 2023-08-04 CN disclosed
US-11414418-B2 Compounds useful as immunomodulators BRISTOL-MYERS SQUIBB COMPANY (US) 2022-08-16 US disclosed
US-20220112187-A1 PYRAZOLOPYRIDINE AMINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE HOFFMANN-LA ROCHE INC. (US) 2022-04-14 US disclosed
US-9493474-B2 Inhibitors of the renal outer medullary potassium channel MERCK SHARP & DOHME CORP. (US) 2016-11-15 US disclosed
US-20140288042-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME LLC 2014-09-25 US disclosed
EP-2773351-A2 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2014-09-10 EP disclosed
US-20130231327-A1 Substituted Spiro-Amide Compounds GRUENENTHAL GMBH (DE) 2013-09-05 US disclosed
US-8455475-B2 Substituted spiro-amide compounds GRUENENTHAL GMBH (DE) 2013-06-04 US disclosed
WO-2013066718-A2 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2013-05-10 WO disclosed
EP-2411381-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-02-01 EP disclosed
US-20100249095-A1 Substituted Spiro-amide Compounds GRUENENTHAL GMBH (DE) 2010-09-30 US disclosed
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed
WO-2009102537-A1 INHIBITORS OF CHECKPOINT KINASES MERCK & CO., INC. (US) 2009-08-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220112187-A1 PYRAZOLOPYRIDINE AMINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE SSB, KCNJ1, KCNJ11 ALDH1A1 1043/4885HSD17B10 4394/4885NAMPT 2049/4885
US-20130231327-A1 Substituted Spiro-Amide Compounds BDKRB1, BDKRB2, REN ALDH1A1 2086/4885HSD17B10 4072/4885NAMPT 2232/4885
US-20240287091-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS BCL6, BCL6B, BCOR ALDH1A1 512/4885HSD17B10 278/4885NAMPT 3709/4885
US-11414418-B2 Compounds useful as immunomodulators CD74, HLA-DRB1, CD47 ALDH1A1 1130/4885HSD17B10 3503/4885NAMPT 656/4885
US-20250276981-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS BCL6, BCL6B, BCOR ALDH1A1 512/4885HSD17B10 278/4885NAMPT 3709/4885
US-20140288042-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL KCNJ2, KCNJ11, KCNK2 ALDH1A1 1827/4885HSD17B10 3557/4885NAMPT 2670/4885
US-20100249095-A1 Substituted Spiro-amide Compounds BDKRB1, BDKRB2, REN ALDH1A1 2086/4885HSD17B10 4072/4885NAMPT 2232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.