SCHEMBL4856700

SCHEMBL4856700

O=C(O)c1ccc2c(c1)CCC2NC(=O)c1cc(-c2ccncc2)n[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.43
ROCK2 O75116 6/20 0.39
ROCK1 Q13464 4/20 0.39
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
WDR5 P61964 1/20 0.37
LIPG Q9Y5X9 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
MAPK8 P45983 1/20 0.36
TAS1R3 Q7RTX0 2/20 0.35
TAS1R1 Q7RTX1 2/20 0.35
TAS1R2 Q8TE23 1/20 0.35
LRRK2 Q5S007 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854586 0.86 ROCK2 (0.52) GSK3BROCK2ROCK1NPC1RAB9A
SCHEMBL5233935 0.84 ROCK2 (0.40) GSK3BROCK2RAB9ALIPGALDH1A1
SCHEMBL5232508 0.77 MAPK8 (0.55) GSK3BROCK2MAPK8MKNK1MKNK2
SCHEMBL14348317 0.76 GSK3B (0.45) GSK3BROCK2ROCK1NPC1RAB9A
SCHEMBL5233639 0.75 GSK3B (0.52) GSK3BROCK2ROCK1MAPK8MKNK1
SCHEMBL5236116 0.75 GSK3B (0.52) GSK3BROCK2ROCK1MAPK8MKNK2
SCHEMBL4848283 0.74 GSK3B (0.51) GSK3BROCK2ROCK1MAPK8MKNK2
SCHEMBL13986943 0.74 ALDH1A1 (0.53) GSK3BROCK2NPC1RAB9AMKNK1
SCHEMBL14348304 0.74 ALDH1A1 (0.53) GSK3BROCK2NPC1RAB9AMKNK1
SCHEMBL13986936 0.73 MAPK8 (0.51) GSK3BROCK2MAPK8MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7462613-B2 Pyridazinone derivatives as pharmaceuticals and pharmaceutical compositions containing them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-12-09 US disclosed