SCHEMBL4857339

SCHEMBL4857339

CN(C)CCOc1ccc(-c2ccccc2COC(C)(C)C)cc1C=CC(=O)c1ccccc1CN(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HRH1 P35367 1/20 0.37
PTPN1 P18031 2/20 0.35
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
SLC6A9 P48067 2/20 0.35
P2RY1 P47900 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAOB P27338 3/20 0.35
AR P10275 1/20 0.35
HTR7 P34969 1/20 0.34
MAOA P21397 2/20 0.34
TNFRSF1A P19438 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4857332 0.91 KDM4E (0.37) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4847477 0.90 ALDH1A1 (0.40) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4851092 0.89 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4853598 0.88 MAOB (0.41) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4848073 0.87 HTR7 (0.41) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4847450 0.87 SLC6A9 (0.43) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4848106 0.86 SLC6A9 (0.44) ALDH1A1KDM4ESMN1; SMN2HRH1BCHE
SCHEMBL6394376 0.86 HTR7 (0.46) ALDH1A1KDM4ESMN1; SMN2HRH1PTPN1
SCHEMBL4847804 0.85 MAOB (0.42) ALDH1A1KDM4ESMN1; SMN2HRH1SLC6A9
SCHEMBL4854762 0.84 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2HRH1SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed