SCHEMBL485779

SCHEMBL485779

O=C(NC1CCCC1)c1ccc2ccccc2c1C#Cc1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.48
GAA P10253 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNA5 P22460 1/20 0.46
RAB9A P51151 6/20 0.45
NPC1 O15118 5/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
HTT P42858 2/20 0.45
NR1I2 O75469 1/20 0.45
AHR P35869 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 1/20 0.44
LMNA P02545 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
GRM5 P41594 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
EPHX1 P07099 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL486033 0.98 GAA (0.48) DRD4GAAKMT2AKCNA5RAB9A
SCHEMBL485505 0.86 RAB9A (0.52) DRD4KMT2ARAB9ANPC1KDM4E
Bicarbonate SCHEMBL486058 0.84 MAPT (0.52) DRD4KMT2ARAB9ANPC1KDM4E
SCHEMBL485565 0.78 ERAP1 (0.50)
SCHEMBL485597 0.76 CXCR2 (0.60) KDM4E
SCHEMBL485776 0.76 BBOX1 (0.44) KMT2AALDH1A1HTTSMN1; SMN2MAPT
SCHEMBL485777 0.76 BBOX1 (0.44) KMT2AALDH1A1HTTSMN1; SMN2MAPT
SCHEMBL485718 0.74 EGLN1 (0.46) KMT2AHTTSMN1; SMN2MAPTLMNA
SCHEMBL485720 0.74 EGLN1 (0.46) KMT2AHTTSMN1; SMN2MAPTLMNA
SCHEMBL29481000 0.73 NPC1 (0.58) GAAKMT2ARAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836158-B1 FUSED BICYCLIC CARBOXAMIDE DERIVATIVES FOR USE AS CXCR2 INHIBITORS IN THE TREATMENT OF INFLAMMATION SANOFI AVENTIS DEUTSCHLAND (DE) 2012-02-01 EP claimed