Bicarbonate

Bicarbonate

SCHEMBL486033

O=C(NC1CCCC1)c1ccc2ccccc2c1C#Cc1ccc(Cl)cc1.O=C(O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.48
KMT2A Q03164 2/20 0.48
DRD4 P21917 3/20 0.47
KCNA5 P22460 1/20 0.45
RAB9A P51151 3/20 0.44
NPC1 O15118 3/20 0.43
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
HTT P42858 2/20 0.43
NR1I2 O75469 1/20 0.43
AHR P35869 1/20 0.43
MAPT P10636 2/20 0.43
GRM5 P41594 2/20 0.43
RXFP1 Q9HBX9 1/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CNR1 P21554 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL485779 0.98 DRD4 (0.48) GAAKMT2ADRD4KCNA5RAB9A
Bicarbonate SCHEMBL486058 0.87 MAPT (0.52) KMT2ADRD4RAB9ANPC1ALDH1A1
SCHEMBL485505 0.84 RAB9A (0.52) KMT2ADRD4RAB9ANPC1ALDH1A1
SCHEMBL485565 0.78 ERAP1 (0.50)
SCHEMBL485777 0.76 BBOX1 (0.44) KMT2AALDH1A1SMN1; SMN2HTTMAPT
SCHEMBL485597 0.76 CXCR2 (0.60) KDM4E
SCHEMBL485776 0.76 BBOX1 (0.44) KMT2AALDH1A1SMN1; SMN2HTTMAPT
SCHEMBL485720 0.74 EGLN1 (0.46) KMT2ASMN1; SMN2HTTMAPTLMNA
SCHEMBL485718 0.74 EGLN1 (0.46) KMT2ASMN1; SMN2HTTMAPTLMNA
SCHEMBL29481000 0.71 NPC1 (0.58) GAAKMT2ARAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836158-B1 FUSED BICYCLIC CARBOXAMIDE DERIVATIVES FOR USE AS CXCR2 INHIBITORS IN THE TREATMENT OF INFLAMMATION SANOFI AVENTIS DEUTSCHLAND (DE) 2012-02-01 EP claimed