SCHEMBL4857993

SCHEMBL4857993

O=C(CN1CCN(CC(O)COc2ccccc2F)CC1)NC1CCCCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
HPGD P15428 1/20 0.51
SCN5A Q14524 2/20 0.50
SCN1A P35498 1/20 0.50
SCN9A Q15858 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
ADRB2 P07550 1/20 0.50
ADRB1 P08588 1/20 0.50
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
ADRA1A P35348 1/20 0.50
DRD3 P35462 1/20 0.50
HTR2B P41595 1/20 0.50
KCNH2 Q12809 1/20 0.50
LMNA P02545 1/20 0.49
BLM P54132 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4857823 0.99 ALDH1A1 (0.55) ALDH1A1HPGDSCN5ASCN1ASCN9A
SCHEMBL4867392 0.88 SCN5A (0.65) ALDH1A1HPGDSCN5ASCN1ASCN9A
SCHEMBL4865310 0.87 MEN1 (0.56) ALDH1A1HPGDSCN5ASCN1ASCN9A
SCHEMBL4867409 0.87 SCN5A (0.66) ALDH1A1HPGDSCN5ASCN1ASCN9A
SCHEMBL3829686 0.80 ALDH1A1 (0.54) ALDH1A1CYP3A4CYP2D6TSHR
SCHEMBL4865295 0.80 NPSR1 (0.55) ALDH1A1SCN5ACYP3A4CYP2D6TSHR
SCHEMBL16783974 0.79 SCN1A (0.66) SCN5ASCN1ASCN9ACYP2D6KCNH2
SCHEMBL16783976 0.79 SCN1A (0.66) SCN5ASCN1ASCN9ACYP2D6KCNH2
SCHEMBL3831166 0.79 ALDH1A1 (0.53) ALDH1A1CYP3A4
SCHEMBL16784017 0.79 SCN1A (0.66) SCN5ASCN1ASCN9ACYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7407960-B2 Substituted heterocyclic compounds CV THERAPEUTICS, INC. (US) 2008-08-05 US disclosed
US-20070004751-A1 Substituted heterocyclic compounds ELZEIN ELFATIH 2007-01-04 US disclosed
US-7125876-B2 Substituted heterocyclic compounds CV THERAPEUTICS, INC. (US) 2006-10-24 US disclosed
EP-1567525-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2005-08-31 EP disclosed
US-20040152890-A1 Substituted heterocyclic compounds CV THERAPEUTICS, INC. 2004-08-05 US disclosed
WO-2004052887-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2004-06-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040152890-A1 Substituted heterocyclic compounds KCNH1, SDHA, COQ8A ALDH1A1 245/4885HPGD 219/4885SCN5A 26/4885
US-20070004751-A1 Substituted heterocyclic compounds KCNH1, SDHA, COQ8A ALDH1A1 281/4885HPGD 224/4885SCN5A 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.