SCHEMBL4859376

SCHEMBL4859376

CC(C)(C)OC(=O)N1CCN(Cc2ccc3cn(-c4ccccc4[N+](=O)[O-])nc3n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 1/20 0.40
MET P08581 1/20 0.39
KDM4E B2RXH2 2/20 0.39
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
DRD4 P21917 1/20 0.38
TP53 P04637 1/20 0.38
THRB P10828 1/20 0.38
ENPP2 Q13822 1/20 0.38
P2RX3 P56373 1/20 0.37
CTSB P07858 1/20 0.37
KMT2A Q03164 1/20 0.37
ACKR3 P25106 1/20 0.37
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30998112 0.75 MAPT (0.63) ALDH1A1LMNAMAPTMETENPP2
SCHEMBL4435451 0.75 MAPT (0.63) ALDH1A1LMNAMAPTMETENPP2
SCHEMBL219576 0.72 ACKR3 (0.41) ALDH1A1LMNAMAPTMETKDM4E
SCHEMBL14607762 0.71 TERT (0.41) ALDH1A1LMNAMAPTMETKDM4E
SCHEMBL3025284 0.71 ALDH1A1 (0.45) ALDH1A1LMNAMAPTMETKDM4E
SCHEMBL18658168 0.70 VEGFA (0.52) ALDH1A1LMNAMAPTMETKDM4E
SCHEMBL26603989 0.70 ALDH1A1 (0.49) ALDH1A1LMNAMAPTKDM4ECHRM2
SCHEMBL221302 0.69 KMT2A (0.42) ALDH1A1LMNAMAPTTP53KMT2A
SCHEMBL23922807 0.69 GRM5 (0.51) ALDH1A1KDM4ECHRM2CHRM4CHRM1
SCHEMBL617183 0.69 FAAH (0.47) ALDH1A1MAPTKDM4ECHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910380-A1 OXAZOLOPYRIDINE DERIVATIVES AS SIRTUIN MODULATORS Sirtris Pharmaceuticals, Inc. (US) 2008-04-16 EP disclosed
WO-2007019417-A1 OXAZOLOPYRIDINE DERIVATIVES AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2007-02-15 WO disclosed