SCHEMBL4861222

SCHEMBL4861222

CC(O)CONC(=O)c1ccc(F)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.44
CHRNG P07510 1/20 0.44
CHRNB1 P11230 1/20 0.44
CHRNB2 P17787 1/20 0.44
SLC6A2 P23975 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CHRND Q07001 1/20 0.44
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
TAS1R3 Q7RTX0 2/20 0.42
TAS1R1 Q7RTX1 2/20 0.42
KCNQ3 O43525 3/20 0.41
KCNQ2 O43526 3/20 0.41
TAS1R2 Q8TE23 1/20 0.41
ALDH1A1 P00352 1/20 0.41
DPP4 P27487 1/20 0.41
MEN1 O00255 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853536 0.87 TAS1R3 (0.44) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL4856514 0.85 CES2 (0.40) CES2CES1TAS1R3TAS1R1ALDH1A1
SCHEMBL5396300 0.79 CES2 (0.43) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL4859235 0.79 CES2 (0.46) CES2CES1TAS1R3TAS1R1KCNQ3
SCHEMBL5395452 0.79 TRPA1 (0.46) CES2CES1TAS1R3TAS1R1KCNQ3
SCHEMBL5384518 0.78 CHRNA1 (0.49) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL6292243 0.77 MAPK1 (0.46) CES2CES1MAP2K1KCNH2
SCHEMBL4851736 0.77 CHRNA1 (0.44) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL30184258 0.76 RAB9A (0.57) ALDH1A1KMT2ARAB9ANPC1GAA
SCHEMBL5379829 0.76 CES2 (0.53) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7411001-B2 Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids WARNER-LAMBERT COMPANY (US) 2008-08-12 US disclosed
US-20050176820-A1 Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids WARNER-LAMBERT COMPANY 2005-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176820-A1 Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids CYP4X1, CYP2A7, CYP4B1 CHRNA1 2335/4885CHRNG 2503/4885CHRNB1 2816/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.