SCHEMBL486253

SCHEMBL486253

Cc1[nH]n(-c2ccccc2)c(=O)c1C1(C(F)(F)F)C(=O)N(c2ccc(F)cc2)C2=C1C(=O)CC(C)(C)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ELOVL6 Q9H5J4 18/20 1.00
HTT P42858 1/20 1.00
MEN1 O00255 1/20 0.91
KMT2A Q03164 1/20 0.91
ELOVL3 Q9HB03 6/20 0.88
MAPT P10636 1/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL486064 1.00 ELOVL6 (1.00) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486051 0.95 ELOVL6 (1.00) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486655 0.94 ELOVL6 (1.00) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486406 0.93 ELOVL6 (0.91) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486256 0.93 ELOVL6 (0.91) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486551 0.92 ELOVL6 (1.00) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486337 0.92 ELOVL6 (1.00) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486069 0.91 ELOVL6 (0.88) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486264 0.91 ELOVL6 (0.86) ELOVL6HTTMEN1KMT2AELOVL3
SCHEMBL486197 0.91 ELOVL6 (0.86) ELOVL6HTTMEN1KMT2AELOVL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106086-B2 Indoledione derivative MSD K.K. (JP) 2012-01-31 US claimed
US-20100056597-A1 INDOLEDIONE DERIVATIVE MSD K.K. (JP) 2010-03-04 US claimed
EP-2145884-A1 INDOLEDIONE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-01-20 EP claimed
EP-2145884-B1 INDOLEDIONE DERIVATIVE MSD KK (JP) 2014-08-06 EP disclosed
US-8106086-B2 Indoledione derivative MSD K.K. (JP) 2012-01-31 US disclosed
US-20100056597-A1 INDOLEDIONE DERIVATIVE MSD K.K. (JP) 2010-03-04 US disclosed
EP-2145884-A1 INDOLEDIONE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-01-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056597-A1 INDOLEDIONE DERIVATIVE LIPE, IDO1, ADRA1A ELOVL6 1113/4885HTT 212/4885MEN1 2086/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.