SCHEMBL4868155

SCHEMBL4868155

NC(=O)c1cc(S(=O)(=O)N(CO)CCO)sc1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA13 Q8N1Q1 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
VCAM1 P19320 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31
MMP1 P03956 1/20 0.31
MMP7 P09237 1/20 0.31
MMP8 P22894 1/20 0.31
MMP12 P39900 1/20 0.31
MMP13 P45452 1/20 0.31
CHEK1 O14757 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1939622 0.94 VCAM1 (0.37) CA2CA12CA1CA3CA4
SCHEMBL1939205 0.84 GSTO1 (0.42) CA2CA12CA1CA3CA4
SCHEMBL1938623 0.77 VCAM1 (0.40) CA2VCAM1SMN1; SMN2GSTO1
SCHEMBL1938333 0.73 CA2 (0.47) CA2CA12CA1CA3CA4
SCHEMBL1938337 0.72 GSTO1 (0.39) CA2CA12CA1CA3CA4
SCHEMBL1940129 0.69 KDM4E (0.37) CA2CA12CA1CA3CA4
SCHEMBL1940985 0.69 CFTR (0.35) CA2CA12CA1CA3CA4
SCHEMBL1940126 0.69 PSEN1 (0.35) CA2CA12CA1CA3CA4
SCHEMBL1939353 0.69 VCAM1 (0.58) VCAM1SMN1; SMN2
SCHEMBL1939691 0.68 ALDH1A1 (0.49) CA2CA12CA9CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008530042-A 2008-08-07 JP claimed
EP-1851225-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2007-11-07 EP claimed
WO-2006084634-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-08-17 WO claimed
EP-1851225-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2007-11-07 EP disclosed
WO-2006084634-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-08-17 WO disclosed