SCHEMBL4872659

SCHEMBL4872659

CCOC(=O)C(CCC(=O)NC(c1ccccc1)(c1ccccc1)c1ccccc1)CP(=O)(O)Cc1ccc2c(c1)C(C)(C)CC2(C)C

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.37
MMP1 P03956 12/20 0.37
MMP13 P45452 11/20 0.35
MMP3 P08254 4/20 0.35
MMP2 P08253 4/20 0.35
MMP8 P22894 2/20 0.35
MMP12 P39900 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27615261 0.79 SMN1; SMN2 (0.42) HSD17B10MMP8
SCHEMBL4872670 0.78 KDM4E (0.31) HSD17B10
SCHEMBL4872665 0.78
SCHEMBL4874698 0.72 FOLH1 (0.39)
SCHEMBL4871262 0.69 MEN1 (0.39) HSD17B10MMP8
SCHEMBL4874207 0.68 CYP26B1 (0.44)
SCHEMBL3516029 0.64 GRM3 (0.40)
SCHEMBL27615259 0.64 SMN1; SMN2 (0.49) HSD17B10MMP1
SCHEMBL31516059 0.64 HSD17B10 (0.53) HSD17B10MMP1MMP13MMP3MMP2
SCHEMBL4872675 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7402576-B2 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2008-07-22 US disclosed
EP-1599487-B1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2007-07-11 EP disclosed
US-20060052616-A1 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2006-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052616-A1 Phosphinic acid analogs of glutamate GLUL, GRIA1, GRM1 HSD17B10 1740/4885MMP1 4142/4885MMP13 4645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.